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Dive into the research topics where Craig R. Woods is active.

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Featured researches published by Craig R. Woods.


Bioorganic & Medicinal Chemistry Letters | 2002

Synthesis and DNA binding properties of saturated distamycin analogues.

Craig R. Woods; Nicolas Faucher; Bernd Eschgfaller; Kenneth W. Bair; Dale L. Boger

A series of saturated heterocyclic analogues of distamycin were prepared and examined. A fluorescent intercalator displacement (FID) assay conducted on p[dA]-p[dT] DNA to obtain C(50) values and a hairpin deoxyoligonucleotide containing an A/T-rich binding site was used to evaluate DNA binding affinity. It is observed that saturated heterocycles greatly reduce the DNA binding relative to distamycin.


Journal of the American Chemical Society | 2002

Hairpin versus extended DNA binding of a substituted β-alanine linked polyamide

Craig R. Woods; Takahiro Ishii; Bing Wu; Kenneth W. Bair; Dale L. Boger


Journal of the American Chemical Society | 2002

Synthesis and DNA binding properties of iminodiacetic acid-linked polyamides: characterization of cooperative extended 2:1 side-by-side parallel binding.

Craig R. Woods; Takahiro Ishii; Dale L. Boger


Archive | 2008

Aryl sulfonamide compounds as modulators of the cck2 receptor

Brett D. Allison; Michael H. Rabinowitz; Mark D. Rosen; Craig R. Woods


Archive | 2014

Quinolinyl modulators of RORγt

Kristi A. Leonard; Kent Barbay; James P. Edwards; Kevin D. Kreutter; David A. Kummer; Umar Maharoof; Rachel Nishimura; Maud Urbanski; Hariharan Venkatesan; Aihua Wang; Ronald L. Wolin; Craig R. Woods; Xiaohua Xue; Maxwell D. Cummings; Kelly J. Mcclure; Virginia M. Tanis


Archive | 2017

moduladores de ror t de quinolinila ligada à heteroarila

Aihua Wang; Anne M. Fourie; Craig R. Woods; David A. Kummer; Hariharan Venkatesan; James P. Edwards; Kent Barbay; Kevin D. Kreutter; Kristi Leonard; Maud Urbanski; Rachel Nishimura; Ronald L. Wolin; Umar Maharoof; Xiaohua Xue


Archive | 2017

6-AMINOPIRIDIN-3-IL TIAZOLES COMO MODULADORES DE RORyT

Steven Goldberg; Mcclure Kelly; Virginia M. Tanis; Elizabeth G Fennema; Alec D. Lebsack; Connor L Martin; Venkatesan Hariharan; Xue Xiaohua; Craig R. Woods


Archive | 2014

Modulateurs quinolinyl à liaison alkyle de ror(gamma)t

Kristi Leonard; Kent Barbay; James P. Edwards; Kevin D. Kreutter; David A. Kummer; Umar Maharoof; Rachel Nishimura; Maud Urbanski; Hariharan Venkatesan; Aihua Wang; Ronald L. Wolin; Craig R. Woods; Anne M. Fourie; Xiaohua Xue; Maxwell D. Cummings


Archive | 2013

Modulateurs de ror-gamma-t de type quinolinyle à liaison méthylène

Kristi Leonard; Kent Barbay; James P. Edwards; Kevin D. Kreutter; David A. Kummer; Umar Maharoof; Rachel Nishimura; Maud Urbanski; Hariharan Venkatesan; Aihua Wang; Ronald L. Wolin; Craig R. Woods; Joan Pierce; Steven Goldberg; Anne M. Fourie; Xiaohua Xue


Bioorganic & Medicinal Chemistry Letters | 2010

Corrigendum to Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2α (HRI) kinase

Mark D. Rosen; Craig R. Woods; Steven Goldberg; Michael D. Hack; A. Dawn Bounds; Young Yang; Pamela C. Wagaman; Victor K. Phuong; Angela P. Ameriks; Terrance D. Barrett; Kimon C. Kanelakis; Jui Chang Chuang; Nigel P. Shankley; Michael H. Rabinowitz

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Aihua Wang

University of Science and Technology

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Dale L. Boger

Scripps Research Institute

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