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Dive into the research topics where David A. Mareska is active.

Publication


Featured researches published by David A. Mareska.


Archive | 2009

P38 inhibitors and methods of use thereof

Mark Munson; David A. Mareska; Youngboo Kim; Robert D. Gronenberg; James P. Rizzi; Martha Rodriguez; Ganghyeok Kim; Guy Vigers; Chang Rao; Devan Balachari; Darren Harvey


Bioorganic & Medicinal Chemistry Letters | 2007

Tetrazole and ester substituted tetrahydoquinoxalines as potent cholesteryl ester transfer protein inhibitors.

C. Todd Eary; Zachary Jones; Robert Groneberg; Laurence E. Burgess; David A. Mareska; Mark Drew; James F. Blake; Ellen R. Laird; Devan Balachari; Michael O’Sullivan; Andrew Allen; Vivienne Marsh


Journal of Medicinal Chemistry | 2007

Potent Nonpeptide Antagonists of the Bradykinin B1 Receptor: Structure−Activity Relationship Studies with Novel Diaminochroman Carboxamides

Kaustav Biswas; Aiwen Li; Jian Jeffrey Chen; Derin C. D'amico; Christopher Fotsch; Nianhe Han; Jason Brooks Human; Qingyian Liu; Mark H. Norman; Bobby Riahi; Chester Chenguang Yuan; Hideo Suzuki; David A. Mareska; James Zhan; David E. Clarke; Andras Toro; Robert Groneberg; Laurence E. Burgess; Dianna Lester-Zeiner; Gloria Biddlecome; Barton H. Manning; Leyla Arik; Hong Dong; Ming Huang; Augustus Kamassah; Richard J. Loeloff; Hong Sun; Feng-Yin Hsieh; Gondi Kumar; Gordon Ng


Archive | 2004

Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof

Robert D. Groneberg; Ben Askew; Derin C. D'amico; James Zhan; Andras Toro; Hideo Suzuki; David A. Mareska; Nianh Han; Christopher Fotsch; Qinglan Liu; Babak Riahi; Kevin Yang; Aiwan Li; Chester Chenguang Yuan; Kaustav Biswas; Scott Harried; Tom Nguyen; Wenyuan Qian; Jian J. Chen; Rana Nomak


Archive | 2010

Piperidine-containing compounds and use thereof

Martha Rodriguez; David A. Mareska; Jeremy J. Hans; Darren Harvey; Robert Groneberg; Michael O'sullivan


Journal of Medicinal Chemistry | 2007

Identification of a nonpeptidic and conformationally restricted bradykinin B1 receptor antagonist with anti-inflammatory activity

Derin C. D'amico; Toshi Aya; Jason Brooks Human; Christopher Fotsch; Jian Jeffrey Chen; Kaustav Biswas; Bobby Riahi; Mark H. Norman; Christopher A. Willoughby; Randall W. Hungate; Paul J. Reider; Gloria Biddlecome; Dianna Lester-Zeiner; Carlo Van Staden; Eileen Johnson; Augustus Kamassah; Leyla Arik; Judy Wang; Vellarkad N. Viswanadhan; Robert Groneberg; James Zhan; Hideo Suzuki; Andras Toro; David A. Mareska; David E. Clarke; Darren Harvey; Laurence E. Burgess; Ellen R. Laird; Benny C. Askew; Gordon Ng


Bioorganic & Medicinal Chemistry Letters | 2006

A new class of bradykinin 1 receptor antagonists containing the piperidine acetic acid tetralin core

Christopher Fotsch; Gloria Biddlecome; Kaustav Biswas; Jian Jeff Chen; Derin C. D’Amico; Robert Groneberg; Nianhe Bruce Han; Feng-Yin Hsieh; Augustus Kamassah; Gondi Kumar; Dianna Lester-Zeiner; Qingyian Liu; David A. Mareska; Babak Riahi; Yueh-Ju Judy Wang; Kevin Yang; James Zhan; Joe Zhu; Eileen Johnson; Gordon Ng; Benny C. Askew


Archive | 2011

SUBSTITUTED N-(1H-INDAZOL-4-YL)IMIDAZO[1,2-a]PYRIDINE-3-CARBOXAMIDE COMPOUNDS AS TYPE III RECEPTOR TYROSINE KINASE INHIBITORS

Mark Laurence Boys; Robert Kirk Delisle; Erik James Hicken; April L. Kennedy; David A. Mareska; Fredrik P. Marmsater; Mark Munson; Brad Newhouse; Bryson Rast; James P. Rizzi; Martha Rodriguez; George T. Topalov; Qian Zhao


Archive | 2004

P38 inhibitor und anwendungsverfahren dafür

Mark Munson; David A. Mareska; Youngboo Kim; Robert Groneberg; James P. Rizzi; Martha Rodriguez; Ganghyeok Kim; Guy Vigers; Chang Rao; Devan Balachari; Darren Harvey


Archive | 2015

BENZOIMIDAZOL-1,2-YL AMIDES AS Kv7 CHANNEL ACTIVATORS

Lynn Resnick; George T. Topalov; Steven A. Boyd; Justin K. Belardi; Charles A. Flentge; James S. Hale; Scott Harried; David A. Mareska; Kai Zhang

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