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Publication
Featured researches published by Douglas John Jenkins.
ACS Medicinal Chemistry Letters | 2010
Lori Krim Gavrin; Paige Erin Mahaney; Douglas John Jenkins; Lisa M. Nogle; Cheryl A. Mugford; Christine Huselton; Jennifer Leiter; Grace H. Johnston; Jenifer A. Bray; Kevin D. Burroughs; Scott Cosmi; Peter D. Alfinito; Douglas M. Ho; Darlene C. Deecher; Eugene John Trybulski
The potency and selectivity of a series of 1-{(1S)-2-[amino]-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol analogues are described. These compounds were prepared to improve in vitro metabolic stability and achieve brain penetration. Compound 13 (WAY-260022, NRI-022) was found to be a potent inhibitor of norepinephrine reuptake and demonstrated excellent selectivity over the serotonin and dopamine transporters. Additionally, 13 exhibited oral efficacy in a rat model of thermoregulatory dysfunction.
Organic Letters | 2006
Matthew L. Crawley; Igor Goljer; Douglas John Jenkins; John F. Mehlmann; Lisa M. Nogle; Rebecca Dooley; Paige Erin Mahaney
Archive | 2004
Paige Erin Mahaney; Lori Krim Gavrin; Douglas John Jenkins
Archive | 2006
Paige Erin Mahaney; Gavin David Heffernan; Richard D. Coghlan; Stephen Todd Cohn; Callain Younghee Kim; Douglas John Jenkins; Michael Anthony Marella; Casey Cameron Mccomas; Joseph Peter Sabatucci; Eugene A. Terefenko; Eugene John Trybulski; An Thien Vu; Fei Ye; Puwen Zhang
Archive | 2004
Paige Erin Mahaney; Lori Danielle Krim; Douglas John Jenkins
Archive | 2009
Thomas J. Commons; Douglas John Jenkins; Eugene John Trybulski; Andrew Fensome
Archive | 2007
Casey Cameron Mccomas; Stephen Todd Cohn; Matthew L. Crawley; Andrew Fensome; Joel Adam Goldberg; Douglas John Jenkins; Callain Younghee Kim; Paige Erin Mahaney; Charles William Mann; Michael Anthony Marella; David John O'Neill; Joseph Peter Sabatucci; Eugene A. Terefenko; Eugene John Trybulski; An Thien Vu; Richard Page Woodworth; Puwen Zhang
Archive | 2006
Paige Erin Mahaney; Gavin David Heffernan; Richard D. Coghlan; Stephen Todd Cohn; Callain Younghee Kim; Douglas John Jenkins; Michael Anthony Marella; Casey Cameron Mccomas; Joseph Peter Sabatucci; Eugene A. Terefenko; Eugene John Trybulski; An Thien Vu; Fei Ye; Puwen Zhang
Archive | 2006
Paige Erin Mahaney; Gavin David Heffernan; Richard D. Coghlan; Stephen Todd Cohn; Callain Younghee Kim; Douglas John Jenkins; Michael Anthony Marella; Casey Cameron Mccomas; Joseph Peter Sabatucci; Eugene A. Terefenko; Eugene John Trybulski; An Thien Vu; Fei Ye; Puwen Zhang
Archive | 2004
Paige Erin Mahaney; Lori Danielle Krim; Douglas John Jenkins