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Featured researches published by Eiichi Okezaki.


Chemical & Pharmaceutical Bulletin | 2001

Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 2. 1) Relationship between Lipophilicity and Antibacterial Activity in 5-Thiocarbonyl Oxazolidinones

Ryukou Tokuyama; Yoshiei Takahashi; Yayoi Tomita; Masatoshi Tsubouchi; Toshihiko Yoshida; Nobuhiko Iwasaki; Noriyuki Kado; Eiichi Okezaki; Osamu Nagata


Chemical & Pharmaceutical Bulletin | 2001

Structure-Activity Relationship(SAR)Studies on Oxazolidinone Antibacterial Agents.1. Conversion of 5-Substituent on Oxazolidinone

Ryukou Tokuyama; Yoshiei Takahashi; Yayoi Tomita; Tomio Suzuki; Toshihiko Yoshida; Nobuhiko Iwasaki; Noriyuki Kado; Eiichi Okezaki; Osamu Nagata


Chemical & Pharmaceutical Bulletin | 2001

Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 3. 1) Synthesis and Evaluation of 5-Thiocarbamate Oxazolidinones

Ryukou Tokuyama; Yoshiei Takahashi; Yayoi Tomita; Masatoshi Tsubouchi; Nobuhiko Iwasaki; Noriyuki Kado; Eiichi Okezaki; Osamu Nagata


Journal of pharmacobio-dynamics | 1988

Entry of the New Quinolone Antibacterial Agents of Ofloxacin and NY-198 into the Central Nervous System in Rats

Hitoshi Sato; Eiichi Okezaki; Setsuko Yamamoto; Osamu Nagata; Hideo Kato; Akira Tsuji


Journal of Pharmaceutical Sciences | 1989

Serum Protein Binding of Lomefloxacin, a New Antimicrobial Agent, and Its Related Quinolones

Eiichi Okezaki; Tetsuya Terasaki; Masato Nakamura; Osamu Nagata; Hideo Kato; Akira Tsuji


Journal of Antimicrobial Chemotherapy | 1997

In-vitro antimicrobial activity of HSR-903, a new fluoroquinolone, against clinical isolates of Neisseria gonorrhoeae with quinolone resistance-associated alterations in GyrA and ParC.

Takashi Deguchi; Mitsuru Yasuda; Satoshi Ishihara; Yoshie Takahashi; Eiichi Okezaki; Osamu Nagata; Isao Saito; Yukimichi Kawada


Chemical & Pharmaceutical Bulletin | 1988

Kinetic Analysis of the Peritoneal Transport of Quinolonecarboxylic Acids in Rats

Hitoshi Sato; Fusashi Ishikawa; Eiichi Okezaki; Osamu Nagata; Emi Nakashima; Yoshiharu Deguchi; Fujio Ichimura; Akira Tsuji


Chemical & Pharmaceutical Bulletin | 1984

Sparsomycin Analogs. III. Synthesis and Biological Activities of (E)-β-(6-Methyluracil-5-yl) acrylic Acid Derivatives

Shoichi Kanatomo; Sotoo Nagai; Kazuhiro Ohki; Tetsuko Hase; Chiaki Nomura; Eiichi Okezaki


Chemotherapy | 2004

Subject Index Vol. 50, 2004

Satoshi Yoshizumi; Yoshie Takahashi; Yoshinari Watanabe; Eiichi Okezaki; Yoshikazu Ishii; Kazuhiro Tateda; F. Meyer; A. Lueck; A. Hribaschek; H. Lippert; K. Ridwelski; Tetsuya Oguri; Carrillo-Muñoz Aj; A. Guglietta; Constantinos L. Petrogiannopoulos; Sotirios G. Kalogeropoulos; Dimitrios C. Dandakis; Georgios A. Hartzoulakis; George N. Karahalios; Christos P. Flevaris; Antonios K. Zacharof; Hiroyuki Achiwa; Daisuke Kato; Hiroyoshi Maeda; Takashi Niimi; Shigeki Sato; Ryuzo Ueda; A. Lale Doğan; Ayça Doğan; Hande Canpinar


Journal of Toxicologic Pathology | 1998

Significance of Intraglomerular Expression of α-Smooth Muscle Actin, Desmin, and PDGF Receptor on Glomerulosclerosis in the Rat Remnant Kidney Model

Takeo Shimo; Masafumi Ohshita; Junichi Katayama; Akemi Saito; Yasuji Aoki; Eiichi Okezaki; Osamu Nagata

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Nobuhiko Iwasaki

Tokyo Medical and Dental University

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