Network


Latest external collaboration on country level. Dive into details by clicking on the dots.

Hotspot


Dive into the research topics where Fabrice Vergne is active.

Publication


Featured researches published by Fabrice Vergne.


Archive | 2005

3- or 4-monosubstituted phenol and thiophenol derivatives useful as H3 ligands

Patrick Bernardelli; Andrew Michael Cronin; Alexis Denis; Stephen Martin Denton; Henry Jacobelli; Mark Ian Kemp; Edwige Lorthiois; Fiona Rousseau; Delphine Serradeil-Civit; Fabrice Vergne


Bioorganic & Medicinal Chemistry Letters | 2004

Discovery of thiadiazoles as a novel structural class of potent and selective PDE7 inhibitors. Part 1: Design, synthesis and structure–activity relationship studies

Fabrice Vergne; Patrick Bernardelli; Edwige Lorthiois; Nga Pham; Emmanuelle Proust; Chrystelle Oliveira; Abdel-Kader Mafroud; Frederique Royer; Roger Wrigglesworth; Jennifer K. Schellhaas; Mark Robert Barvian; François Moreau; Moulay Idrissi; Anita Tertre; Bernadette Bertin; Magali Coupe; Patrick Berna; Patricia Soulard


Archive | 2002

Spirotricyclic derivatives and their use as phosphodiesterase-7 inhibitors

Patrick Bernardelli; Pierre Ducrot; Edwige Lorthiois; Fabrice Vergne


Archive | 2003

Spirocondensed quinazolinones and their use as phosphodiesterase inhibitors

Patrick Bernardelli; Fabrice Vergne; Chrystelle Uk Patent Dept Pfizer Limted Mendes; Pierre Ducrot


Bioorganic & Medicinal Chemistry Letters | 2004

Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 1

Edwige Lorthiois; Patrick Bernardelli; Fabrice Vergne; Chrystelle Oliveira; Abdel-Kader Mafroud; Emmanuelle Proust; Lamia Heuze; François Moreau; Moulay Idrissi; Anita Tertre; Bernadette Bertin; Magali Coupe; Roger Wrigglesworth; Arnaud Descours; Patricia Soulard; Patrick Berna


Bioorganic & Medicinal Chemistry Letters | 2004

Discovery of thiadiazoles as a novel structural class of potent and selective PDE7 inhibitors. Part 2: Metabolism-directed optimization studies towards orally bioavailable derivatives

Fabrice Vergne; Patrick Bernardelli; Edwige Lorthiois; Nga Pham; Emmanuelle Proust; Chrystelle Oliveira; Abdel-Kader Mafroud; Pierre Ducrot; Roger Wrigglesworth; Françoise Berlioz-Seux; Francis Coleon; Eric Chevalier; François Moreau; Moulay Idrissi; Anita Tertre; Arnaud Descours; Patrick Berna; Mei Li


Bioorganic & Medicinal Chemistry Letters | 2004

Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 2: Optimization of 5,8-disubstituted derivatives

Patrick Bernardelli; Edwige Lorthiois; Fabrice Vergne; Chrystelle Oliveira; Abdel-Kader Mafroud; Emmanuelle Proust; Nga Pham; Pierre Ducrot; François Moreau; Moulay Idrissi; Anita Tertre; Bernadette Bertin; Magali Coupe; Eric Chevalier; Arnaud Descours; Françoise Berlioz-Seux; Patrick Berna; Mei Li


Archive | 2001

Thiadiazoles and oxadiazoles and their use as phosphodiesterase-7 inhibitors

Fabrice Vergne; Pierre Ducrot; Charles Andrianjara; Patrick Bernardelli; Edwige Lorthois


Annual Reports in Medicinal Chemistry | 2005

PDE7 Inhibitors: Chemistry and Potential Therapeutic Utilites

Fabrice Vergne; Patrick Bernardelli; Eric Chevalier


Archive | 2003

(4,2-Disubstituted-thiazol-5-yl)amine compounds as PDE7 inhibitors

Fabrice Vergne; Patrick Bernardelli; Edwige Lorthiois; Pierre Ducrot

Researchain Logo
Decentralizing Knowledge