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Dive into the research topics where Francois Audiau is active.

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Featured researches published by Francois Audiau.


Synthetic Communications | 1992

Versatile Methods for the Synthesis of 2-Amino-6-trifluoromethoxy-(nitro)benzothiazoles

Serge Mignani; Francois Audiau; Joseph Le Blevec; Conception Nemecek; Michel Barreau; Patrick Jimonet; Claude Gueremy

Abstract Convenient and regioselective syntheses of all three isomers of mononitro-6-trifluoromethoxy-benzothiazoles, starting from 2-amino-6-trifluoromethoxy-benzothiazole (riluzole) are described.


Journal of Medicinal Chemistry | 1999

Riluzole Series. Synthesis and in Vivo “Antiglutamate” Activity of 6-Substituted-2-benzothiazolamines and 3-Substituted-2-imino-benzothiazolines

Patrick Jimonet; Francois Audiau; Michel Barreau; Jean-Charles Blanchard; Alain Boireau; Yvette Bour; Marie-Annick Coléno; Adam Doble; Gilles Doerflinger; Claudine Do Huu; Marie-Hélène Donat; Jean Marie Duchesne; Pierre Ganil; Claude Gueremy; Eliane Honoré; Bernard Just; Roselyne Kerphirique; Sylvie Gontier; Philippe Hubert; Pierre M. Laduron; Joseph Le Blevec; Mireille Meunier; Jean-Marie Miquet; Conception Nemecek; Martine Pasquet; Odile Piot; Jeremy Pratt; Jean Rataud; Michel Reibaud; and Jean-Marie Stutzmann


Archive | 1994

7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS

Jean-Claude Aloup; Francois Audiau; Dominique Damour; Arielle Genevois-Borella; Patrick Jimonet; Serge Mignani


Archive | 1993

3,4-DIHYDRO-2H-1,2,4-BENZOTHIADIAZINE-1,1-DIOXIDE-3-CARBOXYLIC ACID DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME.

Jean-Claude Aloup; Francois Audiau; Dominique Damour; Patrick Jimonet; Serge Mignani


Archive | 1994

IMIDAZO[1,2-a]PYRAZINE-4-ONE, PREPARATION THEREOF AND DRUGS CONTAINING SAME

Jean-Claude Aloup; Francois Audiau; Dominique Damour; Arielle Genevois-Borella; Patrick Jimonet; Serge Mignani; Yves Ribeill


Archive | 1989

Medicaments containing 2-benzothiazolamine derivatives, compounds and their preparation

Francois Audiau; Claude James


Archive | 1991

Pharmaceutical compositions, 2-benzothiazolamine derivatives, and their preparation

Francois Audiau; Claude James


Journal of Medicinal Chemistry | 1980

3-(4-Piperidinylalkyl)indoles, selective inhibitors of neuronal 5-hydroxytryptamine uptake.

Claude Gueremy; Francois Audiau; Alain Champseix; Andre Uzan; Gérard Le Fur; Jean Rataud


Archive | 1995

5h-indeno[1,2-b]pyrazine-2,3-dione derivatives, preparation thereof and drugs containing same

Jean-Claude Aloup; Francois Audiau; Michel Barreau; Dominique Damour; Arielle Genevois-Borella; Patrick Jimonet; Serge Magnani; Yves Ribeill


Archive | 1995

INDENO[1,2-e]PYRAZINE-4-ONES, PREPARATION THEREOF AND DRUGS CONTAINING SAME

Jean-Claude Aloup; Francois Audiau; Michel Barreau; Dominique Damour; Arielle Genevois-Borella; Patrick Jimonet; Serge Mignani; Yves Ribeill

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