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Dive into the research topics where Hideaki Inada is active.

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Featured researches published by Hideaki Inada.


Chemical & Pharmaceutical Bulletin | 2017

Discovery of Peripheral κ-Opioid Receptor Agonists as Novel Analgesics

Shinya Suzuki; Yuji Sugawara; Hideaki Inada; Riichiro Tsuji; Atsushi Inoue; Ryuji Tanimura; Rieko Shimozono; Mitsuhiro Konno; Tomofumi Ohyama; Eriko Higashi; Chizuka Sakai; Koji Kawai

κ-Opioid receptor agonists with high selectivity over the μ-opioid receptor and peripheral selectivity are attractive targets in the development of drugs for pain. We have previously attempted to create novel analgesics with peripheral selective κ-opioid receptor agonist on the basis of TRK-820. In this study, we elucidated the biological properties of 17-hydroxy-cyclopropylmethyl and 10α-hydroxy derivatives. These compounds were found to have better κ-opioid receptor selectivity and peripheral selectivity than TRK-820.


Archive | 1998

Remedies for drug addiction

Hiroshi Nagase; Takashi Endoh; Tsutomu Suzuki; Kuniaki Kawamura; Koji Oshima; Hideaki Inada


Archive | 1999

Antipruritic for cornea or conjunctiva

Hideaki Inada; Kuniaki Kawamura; Hiroshi Nagase; Kiyoshi Okano; Hiroko Togashi; Jun Uchiumi; 潤 内海; 裕子 冨樫; 清 岡野; 邦昭 川村; 英朗 稲田; 長瀬 博


Archive | 2002

Remedies for sepsis

Tomohiko Suzuki; Hideaki Inada; Yoshitaka Yoshizawa; Kuniaki Kawamura; Toshiaki Tanaka


Archive | 2016

Morphinan derivative and medicinal use for same

理一郎 辻; Riichiro Tsuji; 孝治 河合; Koji Kawai; 英朗 稲田; Hideaki Inada; 雄二 菅原; Yuji Sugawara


Archive | 2016

Dérivé de morphinane et son usage médical

理一郎 辻; Riichiro Tsuji; 孝治 河合; Koji Kawai; 英朗 稲田; Hideaki Inada; 雄二 菅原; Yuji Sugawara


Archive | 2002

Mittel zur behandlung von sepsis

Tomohiko Suzuki; Hideaki Inada; Yoshitaka Yoshizawa; Kuniaki Kawamura; Toshiaki Tanaka


Archive | 2002

Therapeutic agent for sepsis

Tomohiko Suzuki; Hideaki Inada; Yoshitaka Yoshizawa; Kuniaki Kawamura; Toshiaki Tanaka


Archive | 1998

Remedes contre la toxicomanie

Hiroshi Nagase; Takashi Endoh; Tsutomu Suzuki; Kuniaki Kawamura; Koji Oshima; Hideaki Inada


Archive | 1998

PHARMACEUTICAL COMPOSITION CONTAINING MORPHINAN DERIVATIVE FOR TREATING DRUG DEPENDENCE

Hiroshi Nagase; Takashi Endoh; Tsutomu Suzuki; Kuniaki Kawamura; Koji Oshima; Hideaki Inada

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Hiroshi Nagase

Medical College of Wisconsin

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