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Dive into the research topics where Itaru Tsukada is active.

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Featured researches published by Itaru Tsukada.


Bioorganic & Medicinal Chemistry Letters | 2010

Synthesis and evaluation of novel antifungal agents-quinoline and pyridine amide derivatives

Kazutaka Nakamoto; Itaru Tsukada; Keigo Tanaka; Masayuki Matsukura; Toru Haneda; Satoshi Inoue; Norio Murai; Shinya Abe; Norihiro Ueda; Mamiko Miyazaki; Naoaki Watanabe; Makoto Asada; Kentaro Yoshimatsu; Katsura Hata

Quinoline amide, azaindole amide and pyridine amides were synthesized and tested for in vitro antifungal activity against fungi. These synthesized amides have potent antifungal activity against Candida albicans and Aspergillus fumigatus. Our results suggest that hetero ring amides may be potent antifungal agents that operate by inhibiting the function of Gwt1 protein in the GPI biosynthetic pathway.


Archive | 1996

Preventing and therapeutic agent for viral infectious disease

Yasunobu Kai; Yumiko Kako; Manabu Sasho; Itaru Tsukada; Manabu Yanagisawa; 学 佐生; 由美子 加来; 格 塚田; 学 柳澤; 康信 甲斐


Archive | 2002

2-iminopyrrolidine derivatives

Shuichi Suzuki; Makoto Kotake; Mitsuaki Miyamoto; Tetsuya Kawahara; Akiharu Kajiwara; Ieharu Hishinuma; Kazuo Okano; Syuhei Miyazawa; Richard Clark; Fumihiro Ozaki; Nobuaki Sato; Masanobu Shinoda; Atsushi Kamada; Itaru Tsukada; Fumiyoshi Matsuura; Yoshimitsu Naoe; Taro Terauchi; Yoshiaki Oohashi; Osamu Ito; Hiroshi Tanaka; Takashii Musha; Motoji Kogushi; Tsutomu Kawata; Toshiyuki Matsuoka; Hiroko Kobayashi; Keni-ichi Chiba; Akifumi Kimura; Naoto Ono


Archive | 2004

Novel antifungal agent comprising heterocyclic compound

Kazutaka Nakamoto; Itaru Tsukada; Keigo Tanaka; Masayuki Matsukura; Toru Haneda; Satoshi Inoue; Norihiro Ueda; Shinya Abe; Katsura Hata; Naoaki Watanabe


Chemical & Pharmaceutical Bulletin | 1998

Synthesis and antifungal activity of novel thiazole-containing triazole antifungals. II. Optically active ER-30346 and its derivatives.

Akihiko Tsuruoka; Yumiko Kaku; Hiroyuki Kakinuma; Itaru Tsukada; Manabu Yanagisawa; Kazumasa Nara; Toshihiko Naito


Archive | 2008

Fungal cell wall synthesis gene

Kappei Tsukahara; Katsura Hata; Koji Sagane; Kazutaka Nakamoto; Mamiko Tsuchiya; Naoaki Watanabe; Fuminori Ohba; Itaru Tsukada; Norihiro Ueda; Keigo Tanaka; Junko Kai


Archive | 2002

2-iminoimidazole derivatives (2)

Shuichi Suzuki; Makoto Kotake; Mitsuaki Miyamoto; Tetsuya Kawahara; Akiharu Kajiwara; Ieharu Hishinuma; Kazuo Okano; Syuhei Miyazawa; Richard Clark; Fumihiro Ozaki; Nobuaki Sato; Masanobu Shinoda; Atsushi Kamada; Itaru Tsukada; Fumiyoshi Matsuura; Yoshimitsu Naoe; Taro Terauchi; Yoshiaki Oohashi; Osamu Ito; Hiroshi Tanaka; Takahashi Musha; Motoji Kogushi; Tsutomu Kawata; Toshiyuki Matsuoka; Hiroko Kobayashi; Kenichi Chiba; Akifumi Kimura; Naoto Ono


Archive | 2011

Novel antifungal agent containing heterocyclic compound

Kazutaka Nakamoto; Itaru Tsukada; Keigo Tanaka; Masayuki Matsukura; Toru Haneda; Satoshi Inoue; Norihiro Ueda; Shinya Abe; Katsura Hata; Naoaki Watanabe


Archive | 2005

Novel Antimalarial Agent Containing Heterocyclic Compound

Kazutaka Nakamoto; Masayuki Matsukura; Keigo Tanaka; Satoshi Inoue; Itaru Tsukada; Toru Haneda; Norihiro Ueda; Shinya Abe; Koji Sagane


Archive | 2002

Cyclic amidine derivative

Shuichi Suzuki; Makoto Kotake; Mitsuaki Miyamoto; Tetsuya Kawahara; Akiharu Kajiwara; Ieharu Hishinuma; Kazuo Okano; Syuhei Miyazawa; Richard Clark; Fumihiro Ozaki; Nobuaki Sato; Masanobu Shinoda; Atsushi Kamada; Itaru Tsukada; Fumiyoshi Matsuura; Yoshimitsu Naoe; Taro Terauchi; Yoshiaki Oohashi; Osamu Ito; Hiroshi Tanaka; Takashi Musha; Motoji Kogushi; Tsutomu Kawata; Toshiyuki Matsuoka; Hiroko Kobayashi; Kenichi Chiba; Akifumi Kimura; Naoto Ono

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