Is this you? Create Your Porfile
Avatar

James J. Droste

Eli Lilly and Company

Network

Latest external collaboration on country level. Dive into details by clicking on the dots.

Explore More

Hotspot

Dive into the research topics where James J. Droste is active.

Explore More

Publication

Featured researches published by James J. Droste.

Tetrahedron Letters | 1996

A diastereoselective tandem metalloenamine alkylation/aza-annulation of β-tetralones expedites the synthesis of benzoquinolinones

James E. Audia; James J. Droste; James M. Dunigan; John L Bowers; Perry Clark Heath; Dale W. Holme; Jill H. Eifert; Harry A. Kay; Richard D. Miller; Jorge M. Olivares; Thomas F. Rainey; Leland Otto Weigel

Abstract In one operation, metalloenamines derived from R -phenylethylamine (PEA) and a β-tetralone were treated with an electrophile followed by acrylic anhydride. The unpurified lactams were reduced to give 10b-angular benzoquinolinones (BQs).

Journal of Medicinal Chemistry | 1996

Potent, selective tetrahydro-β-carboline antagonists of the serotonin 2B (5HT2B) contractile receptor in the rat stomach fundus

James E. Audia; Deborah Ann Evrard; Gwyn R. Murdoch; James J. Droste; Jeffrey S. Nissen; Kathy W. Schenck; Pawel Fludzinski; Virginia L. Lucaites; David L. Nelson; Marlene L. Cohen

Archive | 1997

Methods and compounds for inhibiting beta-amyloid peptide release and/or its synthesis

James E. Audia; Thomas C. Britton; James J. Droste; Beverly K. Folmer; George W. Huffman; Varghese John; Lee H. Latimer; Thomas Edward Mabry; Jeffrey S. Nissen; Warren J. Porter; Jon K. Reel; Eugene D. Thorsett; Jay S. Tung; Jing Wu; Clark Norman Eid; William Leonard Scott

Archive | 1996

5-substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)-and 3-(piperidin-4-yl)-1h-indoles: new 5-ht1f agonists

James E. Audia; Bruce A. Dressman; James J. Droste; James Erwin Fritz; Stephen W. Kaldor; Daniel James Koch; Joseph H. Krushinski; Jeffrey S. Nissen; Vincent Patrick Rocco; John Mehnert Schaus; Dennis Charles Thompson

Archive | 1995

Tetrahydro-beta-carbolines

James E. Audia; James J. Droste; Deborah Ann Evrard; Pawel Fludzinski; Gwyn L. Murdoch; David L. Nelson

Journal of Organic Chemistry | 1994

Stereoselective Epoxidations and Electrophilic Additions to Partial Ergot Alkaloids and Conformationally-Fixed Styrenes. Experimental and Theoretical Modeling Evidence for the Importance of Torsional Steering as a Stereocontrol Element

Michael J. Martinelli; Barry C. Peterson; Vien V. Khau; Darrell R. Hutchison; M. R. Leanna; James E. Audia; James J. Droste; Yun-Dong Wu; K. N. Houk

Archive | 1995

8-substituted tetrahydro-beta-carbolines

James E. Audia; James J. Droste; Jeffrey S. Nissen

Archive | 1994

Tetrahydro-pyrido-indole

James E. Audia; James J. Droste; Deborah Ann Evrard

Archive | 2002

Heterocyclic compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds

Eugene D. Thorsett; Warren J. Porter; Jeffrey S. Nissen; Lee H. Latimer; James E. Audia; James J. Droste

Journal of Organic Chemistry | 1996

Pictet-Spengler-like Synthesis of Tetrahydro-beta-carbolines under Hydrolytic Conditions. Direct Use of Azalactones as Phenylacetaldehyde Equivalents.

James E. Audia; James J. Droste; Jeffrey S. Nissen; Gwyn L. Murdoch; Deborah Ann Evrard

Explore More

Collaboration

Dive into the James J. Droste's collaboration.

Top Co-Authors
Avatar

James E. Audia

University of South Carolina

View shared research outputs
Top Co-Authors
Avatar

Jeffrey S. Nissen

Eli Lilly and Company

View shared research outputs
Top Co-Authors
Avatar

Eugene D. Thorsett

Eli Lilly and Company

View shared research outputs
Top Co-Authors
Avatar

Lee H. Latimer

Eli Lilly and Company

View shared research outputs
Top Co-Authors
Avatar

Warren J. Porter

Eli Lilly and Company

View shared research outputs
Top Co-Authors
Avatar

Jay S. Tung

Thomas Jefferson University

View shared research outputs
Top Co-Authors
Avatar

Jing Wu

Eli Lilly and Company

View shared research outputs
Top Co-Authors
Avatar

Jon K. Reel

Eli Lilly and Company

View shared research outputs
Top Co-Authors
Avatar

Thomas C. Britton

Eli Lilly and Company

View shared research outputs
Top Co-Authors
Avatar

Thomas Edward Mabry

Eli Lilly and Company

View shared research outputs
Explore More
Researchain Logo
Decentralizing Knowledge