James J. Droste | Researchain

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Tetrahedron Letters | 1996

A diastereoselective tandem metalloenamine alkylation/aza-annulation of β-tetralones expedites the synthesis of benzoquinolinones

James E. Audia; James J. Droste; James M. Dunigan; John L Bowers; Perry Clark Heath; Dale W. Holme; Jill H. Eifert; Harry A. Kay; Richard D. Miller; Jorge M. Olivares; Thomas F. Rainey; Leland Otto Weigel

Abstract In one operation, metalloenamines derived from R -phenylethylamine (PEA) and a β-tetralone were treated with an electrophile followed by acrylic anhydride. The unpurified lactams were reduced to give 10b-angular benzoquinolinones (BQs).

Journal of Medicinal Chemistry | 1996

Potent, selective tetrahydro-β-carboline antagonists of the serotonin 2B (5HT2B) contractile receptor in the rat stomach fundus

James E. Audia; Deborah Ann Evrard; Gwyn R. Murdoch; James J. Droste; Jeffrey S. Nissen; Kathy W. Schenck; Pawel Fludzinski; Virginia L. Lucaites; David L. Nelson; Marlene L. Cohen

Archive | 1997

Methods and compounds for inhibiting beta-amyloid peptide release and/or its synthesis

James E. Audia; Thomas C. Britton; James J. Droste; Beverly K. Folmer; George W. Huffman; Varghese John; Lee H. Latimer; Thomas Edward Mabry; Jeffrey S. Nissen; Warren J. Porter; Jon K. Reel; Eugene D. Thorsett; Jay S. Tung; Jing Wu; Clark Norman Eid; William Leonard Scott

Archive | 1996

5-substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)-and 3-(piperidin-4-yl)-1h-indoles: new 5-ht1f agonists

James E. Audia; Bruce A. Dressman; James J. Droste; James Erwin Fritz; Stephen W. Kaldor; Daniel James Koch; Joseph H. Krushinski; Jeffrey S. Nissen; Vincent Patrick Rocco; John Mehnert Schaus; Dennis Charles Thompson

Archive | 1995