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Dive into the research topics where Jun-ichi Hoshi is active.

Publication


Featured researches published by Jun-ichi Hoshi.


Bioorganic & Medicinal Chemistry Letters | 2004

Synthesis of anilino-monoindolylmaleimides as potent and selective PKCβ inhibitors

Masahiro Tanaka; Shoichi Sagawa; Jun-ichi Hoshi; Fumito Shimoma; Isamu Matsuda; Kenji Sakoda; Tomohiko Sasase; Masanori Shindo; Takashi Inaba


Bioorganic & Medicinal Chemistry | 2006

Synthesis, SAR studies, and pharmacological evaluation of 3-anilino-4-(3-indolyl) maleimides with conformationally restricted structure as orally bioavailable PKCβ-selective inhibitors

Masahiro Tanaka; Shoichi Sagawa; Jun-ichi Hoshi; Fumito Shimoma; Katsutaka Yasue; Minoru Ubukata; Tomoyuki Ikemoto; Yasunori Hase; Mitsuru Takahashi; Tomohiko Sasase; Nobuhisa Ueda; Mutsuyoshi Matsushita; Takashi Inaba


Journal of Medicinal Chemistry | 2005

Synthesis and structure-activity relationships of novel selective factor Xa inhibitors with a tetrahydroisoquinoline ring.

Hiroshi Ueno; Katsuyuki Yokota; Jun-ichi Hoshi; Katsutaka Yasue; Mikio Hayashi; Yasunori Hase; Itsuo Uchida; Kazuo Aisaka; Susumu Katoh; Hidetsura Cho


Archive | 2007

Process for production of 4-oxoquinoline compound

Koji Matsuda; Koji Ando; Shigeji Ohki; Takahiro Yamasaki; Jun-ichi Hoshi


Archive | 2007

Method for producing 4-oxoquinoline compound

Koji Matsuda; Koji Ando; Shigeji Ohki; Jun-ichi Hoshi; Takahiro Yamasaki


Bioorganic & Medicinal Chemistry Letters | 2004

Structure-activity relationships of potent and selective factor Xa inhibitors: benzimidazole derivatives with the side chain oriented to the prime site of factor Xa

Hiroshi Ueno; Susumu Katoh; Katsuyuki Yokota; Jun-ichi Hoshi; Mikio Hayashi; Itsuo Uchida; Kazuo Aisaka; Yasunori Hase; Hidetsura Cho


Bioorganic & Medicinal Chemistry Letters | 2005

Discovery of novel tetrahydroisoquinoline derivatives as potent and selective factor Xa inhibitors.

Hiroshi Ueno; Katsuyuki Yokota; Jun-ichi Hoshi; Katsutaka Yasue; Mikio Hayashi; Itsuo Uchida; Kazuo Aisaka; Yastinori Hase; Susumu Katoh; Hidetsura Cho


Archive | 2006

Process for production of highly pure quinolone compound

Koji Matsuda; Koji Ando; Shigeji Ohki; Takahiro Yamasaki; Jun-ichi Hoshi


Archive | 2007

Procede de production d'un compose 4-oxoquinoline

Koji Matsuda; Koji Ando; Shigeji Ohki; Jun-ichi Hoshi; Takahiro Yamasaki


Archive | 2007

Verfahren zur herstellung einer 4-oxochinolin-verbindung

Koji Matsuda; Koji Ando; Shigeji Ohki; Jun-ichi Hoshi; Takahiro Yamasaki

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