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Dive into the research topics where Kiyoshi Taniguchi is active.

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Featured researches published by Kiyoshi Taniguchi.


Bioorganic & Medicinal Chemistry Letters | 2000

A novel pyridazinone derivative as a nonprostanoid PGI2 agonist.

Kazunori Tsubaki; Kiyoshi Taniguchi; Seiichiro Tabuchi; Osamu Okitsu; Kouji Hattori; Jiro Seki; Kazuo Sakane; Hirokazu Tanaka

A novel optically pure pyridazinone derivative was synthesized and identified as a nonprostanoid PGI2 agonist. It inhibited ADP-induced aggregation of human platelets with an IC50 value of 0.081 microM and has high oral bioavailability (56%) with a long half-life (4.3 h) in rats.


Archive | 1999

Aminoalcohol derivatives and their use as beta 3 adrenergic agonists

Kiyoshi Taniguchi; Minoru Sakurai; Takeshi Kato; Naoaki Fujii; Kenichi Washizuka; Yasuyo Tomishima; Hisashi Takasugi; Yutaka Kohno; Nobuhiro Yamamoto; Naoko Unami; Hirohumi Ishikawa


Archive | 1994

4,5-diaryloxazole derivatives

Kiyoshi Taniguchi; Masanobu Nagano; Kouji Hattori; Kazunori Tsubaki; Osamu Okitsu; Seiichiro Tabuchi


Chemical & Pharmaceutical Bulletin | 1993

Synthesis and antiinflammatory and analgesic properties of 2-amino-1H-benzimidazole and 1,2-dihydro-2-iminocycloheptimidazole derivatives

Kiyoshi Taniguchi; Shinji Shigenaga; Takatomo Ogahara; Takashi Fujitsu; Masaaki Matsuo


Archive | 1996

4,5-diaryl oxazole derivatives

Kiyoshi Taniguchi; Kouji Hattori; Kazunori Tsubaki; Osamu Okitsu; Seiichiro Tabuchi


Archive | 1995

Naphthalene derivatives as prostaglandin i2 agonists

Kiyoshi Taniguchi; Masanobu Nagano; Kouji Hattori; Kazunori Tsubaki; Osamu Okitsu; Seiichiro Tabuchi


Archive | 1993

Substituted acetamide compound

Youichi Shiokawa; Kiyoshi Taniguchi; Kazuhiko Take; Kazunori Tsubaki; Hiroaki Mizuno


Chemical & Pharmaceutical Bulletin | 1985

New 2-Aryliminoimidazolidines. I. Synthesis and Antihypertensive Properties of 2-(2-Phenoxyphenylimino) imidazolidines and Related Compounds

Masaaki Matsuo; Kiyoshi Taniguchi; Yousuke Katsura; Toshiharu Kamitani; Ikuo Ueda


Archive | 1980

2-Imidazoline derivatives, process for the preparation thereof and the pharmaceutical composition of the same

Ukuo Ueda; Masaaki Matsuo; Kiyoshi Taniguchi; Yousuke Katsura


Archive | 1992

ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY

Youichi Shiokawa; Masanobu Nagano; Kiyoshi Taniguchi; Kazuhiko Take; Takeshi Kato; Kazunori Tsubaki

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Takeshi Kato

Takeda Pharmaceutical Company

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