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Archive | 2011

DIHIDRODIAZEPINAS UTILES COMO INHIBIDORES DE PROTEINA QUINASAS.

Kay David; Twin Heather; Damien-Charrier Jean; Knegtel Ronald


Archive | 2018

Pyrazinderivater anvendelige som inhibitorer til ATR kinase

Charrier Jean Damien; Durrant Steven; Kay David; Knegtel Ronald; Maccormick Somhairle; Mortimore Michael; O'donnell Michael; Pinder Joanne; Rutherford Alistair; Virani Anisa Nizarali; Young Stephen; Reaper Philip Michael


Archive | 2018

2-AMINO-6-FLUORO-N-(5-FLUORO-4-(4-(4-(OXETAN-3-YL)PIPERAZINE-1-CARBONYL)PIPERIDIN-1-YL)PYRIDIN-3-YL)PYRAZOLO[1,5ALPHA]PYRIMIDINE-3-CARBOXAMIDE AS INHIBITOR OF ATR KINASE

Ahmad Nadia; Boyall Dean; Charrier Jean-Damien; Davis Chris; Davis Rebecca; Durrant Steven; Etxebarria I Jardi Gorka; Fraysse Damien; Jimenez Juan-Miguel; Kay David; Knegtel Ronald; Middleton Donald; O'donnell Michael; Panesar Maninder; Pierard Francoise; Pinder Joanne; Shaw David; Storck Pierre-Henri; Studley John; Twin Heather


Archive | 2016

COMPOUND USEFUL AS INHIBITOR OF ATR KINASE

Charrier Jean-Damien; Steven Durrant; Kay David; O'donnell Michael; Knegtel Ronald; Somhairle MacCormick; Joanne Pinder; Anisa Nizarali Virani; Young Steven; Haley Binch; Thomas Cleveland; Lev T. D. Fanning; Dennis James Hurley; Pramod Joshi; Urvi Sheth; Alina Silina; Philip Michael Reaper


Archive | 2015

4, 5-DIHYDRO- [1, 2, 4] TRIAZOLO [4,3-F] PTERIDINES AS PROTEIN KINASE PLK1 INHIBITORS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS PLK1 45--[124][43- F]

Charrier Jean-Damien; Kay David; Knegtel Ronald


Archive | 2014

TRICYCLIC PYRAZOLO-PYRIDINE KINASE INHIBITOR

Jimenez Juan-Miguel; John Studley; Knegtel Ronald; Settimo Luca; Davis Chris; Damien Fraysse; Philip N. Collier; Guy Brenchley; Boyall Dean; Miller Andrew; Heather Twin; Young Steven


Archive | 2013

DIHYDRODIAZEPINE USEFUL AS INHIBITOR OF PROTEIN KINASE

Charrier Jean-Damien; Kay David; Knegtel Ronald; Twin Heather


Archive | 2013

2-AMINOPYRIDINE DERIVATIVE USEFUL AS KINASE INHIBITOR

Jimenez Juan-Miguel; Bemis Guy; Maltais Francois; Wang Tiansheng; Knegtel Ronald; Davis Chris; Fraysse Damien; Boyall Dean; Settimo Luca; Young Steven; Mortimore Michael


Archive | 2012

3-Ä2-(3-AZYLAMINO-2-OXO-2H-PYRIDIN-1- YL)ACETYLAMINOÜ-4-OXOPENTANSÄUREDERIVATE UND DEREN VERWENDUNG ALS CASPASE-INHIBITOREN

Charrier Jean-Damien; Knegtel Ronald; Mortimore Michael; Studley John


Archive | 2012

4,5-Dihidro-[1,2,4]triazolo[4,3-F]pteridinas como inhibidores de la proteincinasa PLK1 para el tratamiento de trastornos proliferativos

Charrier Jean-Damien; Kay David; Knegtel Ronald

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Kay David

Vertex Pharmaceuticals

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