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Dive into the research topics where Naoko Matsuura is active.

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Featured researches published by Naoko Matsuura.


Journal of Medicinal Chemistry | 2008

Effect of Cathepsin K Inhibitors on Bone Resorption

Naoki Teno; Keiichi Masuya; Takeru Ehara; Takatoshi Kosaka; Takahiro Miyake; Osamu Irie; Yuko Hitomi; Naoko Matsuura; Ichiro Umemura; Genji Iwasaki; Hiroaki Fukaya; Kazuhiro Toriyama; Noriko Uchiyama; Kazuhiko Nonomura; Ikuo Sugiyama; Motohiko Kometani

On the basis of the pyrrolopyrimidine core structure that was previously discovered, cathepsin K inhibitors having a spiro amine at the P3 have been explored to enhance the target, bone marrow, tissue distribution. Several spiro structures were identified with improved distribution toward bone marrow. The representative inhibitor 7 of this series revealed in vivo reduction in C-terminal telopeptide of type I collagen in rats and monkeys.


Archive | 2004

2,4-di(phenylamino) pyrimidines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders

Carlos Garcia-Echeverria; Takanori Kanazawa; Eiji Kawahara; Keiichi Masuya; Naoko Matsuura; Takahiro Miyake; Osamu Ohmori; Ichiro Umemura


Archive | 2004

2, 4-pyrimidinediamines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders

Carlos Garcia-Echeverria; Takanori Kanazawa; Eiji Kawahara; Keiichi Masuya; Naoko Matsuura; Takahiro Miyake; Osamu Ohmori; Ichiro Umemura; Ruo Steensma; Greg Chopiuk; Jiqing Jiang; Yongqin Wan; Qiang Ding; Qiong Zhang; Nathanael S. Gray; Donald S. Karanewsky


Archive | 2007

Bicyclic derivatives as cetp inhibitors

Masashi Kishida; Naoko Matsuura; Hidetomo Imase; Yuki Iwaki; Ichiro Umemura; Osamu Ohmori; Eiji Kawahara


Bioorganic & Medicinal Chemistry Letters | 2007

Novel scaffold for cathepsin K inhibitors

Naoki Teno; Takahiro Miyake; Takeru Ehara; Osamu Irie; Junichi Sakaki; Osamu Ohmori; Hiroki Gunji; Naoko Matsuura; Keiichi Masuya; Yuko Hitomi; Kazuhiko Nonomura; Miyuki Horiuchi; Keigo Gohda; Atsuko Iwasaki; Ichiro Umemura; Sachiyo Tada; Motohiko Kometani; Genji Iwasaki; Sandra W. Cowan-Jacob; Martin Missbach; Rene Lattmann; Claudia Betschart


Archive | 2003

2,4-diaminopyrimidine derivatives

Rolf Baenteli; Gerhard Zenke; Nigel Graham Cooke; Rudolf O. Duthaler; Gebhard Thoma; Anette Von Matt; Toshiyuki Honda; Naoko Matsuura; Kazuhiko Nonomura; Osamu Ohmori; Ichiro Umemura; Klaus Hinterding; Christos Papageorgiou


Archive | 2006

Pyridinyl amine derivatives as inhibitors of cholesteryl ester transfer protein (cetp)

Junichi Sakaki; Masashi Kishida; Naoko Matsuura; Ichiro Umemura; Eiji Kawahara; Ken Yamada; Kazuhide Konishi; Yuki Iwaki; Hidetomo Imase; Takahiro Miyake


Archive | 2012

El archivo contiene la información técnica propuesta después de la presentación de la solicitud y no se incluye en esta especificación

Rolf Baenteli; Nigel Graham Cooke; Rudolf O. Duthaler; Klaus Hinterding; Toshiyuki Honda; Naoko Matsuura; Kazuhiko Nonomura; Osamu Ohmori; Christos Papageorgiou; Gebhard Thoma; Ichiro Umemura; Matt Anette Von; Gerhard Zenke


Archive | 2008

DERIVADOS BICÍCLICOS COMO INHIBIDORES DE CETP

Masashi Kishida; Naoko Matsuura; Hidetomo Imase; Yuki Iwaki; Ichiro Umemura; Osamu Ohmori; Eiji Kawahara


Archive | 2007

Dérivés bicycliques utilisés comme inhibiteurs de cetp

Masashi Kishida; Naoko Matsuura; Hidetomo Imase; Yuki Iwaki; Ichiro Umemura; Osamu Ohmori; Eiji Kawahara

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