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Archive | 2001

Novel phenylalanine derivatives

Kazuyuki Sagi; Tatsuya Okuzumi; Tatsuhiro Yamada; Shunsuke Kageyama; Yoichiro Shima; Tadakiyo Nakagawa; Munetaka Tokumasu; Masayuki Sugiki; Hajime Ito; Itsuya Tanabe; Tamotsu Suzuki; Akira Nakayama; Kazuyuki Ubukata; Kenji Shinkai; Yasuhiro Tanaka; Misato Noguchi; Ayatoshi Andou; Yoriko Yamamoto; Noriyasu Kataoka; Koichi Fujita


Journal of Medicinal Chemistry | 2003

Rational design, synthesis, and structure-activity relationships of novel factor Xa inhibitors: (2-Substituted-4-amidinophenyl)pyruvic and -propionic acids

Kazuyuki Sagi; Tadakiyo Nakagawa; Masahiro Yamanashi; Shingo Makino; Mitsuo Takahashi; Masaru Takayanagi; Kaoru Takenaka; Nobuyasu Suzuki; Seiji Oono; Noriyasu Kataoka; Kohki Ishikawa; Sayaka Shima; Yumiko Fukuda; Takashi Kayahara; Shunji Takehana; Yoichiro Shima; Kazumi Tashiro; Hiroshi Yamamoto; Ryota Yoshimoto; Seinosuke Iwata; Takashi Tsuji; Kuniya Sakurai; Masataka Shoji


Archive | 2004

Process for producing phenylalanine derivative having quinazolinedione skeleton and intermediate for the same

Noriyasu Kataoka; Akinori Tatara; Masanobu Yatagai; Junko Yamanaka


Archive | 2010

Methods for producing phenylalanine derivatives having a quinazolinedione skeleton and intermediates for production thereof

Noriyasu Kataoka; Akinori Tatara; Masanobu Yatagai; Junko Yamanaka


Archive | 2004

Crystal of phenylalanine derivative and process for producing the same

Shinichiro Takahashi; Noriyasu Kataoka; Akinori Tatara; Toshihiro Matsuzawa


Archive | 2011

METHOD FOR PREPARING PHENYLALANINE DERIVATIVES HAVING QUINAZOLINE-DIONE SKELETON AND INTERMEDIATES FOR USE IN THE PREPARATION OF THE DERIVATIVES

Noriyasu Kataoka; Kotaro Okado; Tatsuhiro Yamada; Koichi Fujita; Tamotsu Suzuki; Tatsuya Okuzumi; Masayuki Sugiki; Akinori Tatara


Archive | 2010

Crystals of phenylalanine derivatives and production methods thereof

Shinichiro Takahashi; Noriyasu Kataoka; Akinori Tatara; Toshihiro Matsuzawa


Archive | 2006

Crystal of phenylalanine derivative, process for producing the same and use thereof

Koichi Fujita; Shinichiro Takahashi; Tatsuya Okuzumi; Tatsuhiro Yamada; Kotaro Okado; Noriyasu Kataoka; Haruko Hirashima; Hideyuki Yamaguchi


Archive | 2006

CRYSTALS OF PHENYLALANINE DERIVATIVES, PRODUCTION METHOD THEREOF AND USE THEREOF

Koichi Fujita; Shinichiro Takahashi; Tatsuya Okuzumi; Tatsuhiro Yamada; Kotaro Okado; Noriyasu Kataoka; Haruko Hirashima; Hideyuki Yamaguchi


Archive | 2010

Crystals of isopropyl ester of N-(2,6-dichlorobenzoyl)-4-[6-(methylamino)methyl-1-methyl-2,4-dioxo-1,4-dihydroquinazoline-3(2H)-yl]-l-phenylalanine hydrochloride, production method thereof and use thereof

Koichi Fujita; Shinichiro Takahashi; Tatsuya Okuzumi; Tatsuhiro Yamada; Kotaro Okado; Noriyasu Kataoka; Haruko Hirashima; Hideyuki Yamaguchi

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