Noriyoshi Yamamoto
SANTEN PHARMACEUTICAL CO., LTD.
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Publication
Featured researches published by Noriyoshi Yamamoto.
Bioorganic & Medicinal Chemistry Letters | 2010
Hiroshi Enomoto; Ayako Sawa; Hiroshi Suhara; Noriyoshi Yamamoto; Hiroyuki Inoue; Chikako Setoguchi; Fumio Tsuji; Masahiro Okamoto; Yoshimasa Sasabuchi; Masato Horiuchi; Masakazu Ban
A three substituted urea derivative, SA13353 (compound 1a), exhibited potent inhibitory activity against lipopolysaccharide (LPS)-induced TNF-alpha production. We focused on the 1,1-substituted moiety (R(1) and R(2)) of SA13353 and investigated substituent effects of this moiety on LPS-induced TNF-alpha production by oral administration in rats. The synthesis of the urea derivatives was performed rapidly in a one-pot manner using a manual synthesizer. Several compounds containing hydrophobic substituents at this moiety showed more potent inhibitory activities than SA13353.
Archive | 2001
Masakazu Ban; Hiroshi Suhara; Masato Horiuchi; Noriyoshi Yamamoto; Hiroshi Enomoto; Hiroyuki Inoue
Archive | 1995
Yoichi Kawashima; Kenichi Fujimura; Hiroshi Suhara; Noriyoshi Yamamoto; Hiromi Matsumoto; Nobuaki Miyawaki; Yuko Fujita
Archive | 1995
Yoichi Kawashima; Kenichi Fujimura; Hiroshi Suhara; Noriyoshi Yamamoto; Hiromi Matsumoto; Nobuaki Miyawaki; Yuko Fujita
Archive | 2012
Kazuhiro Kudou; Noriyoshi Yamamoto; Masakazu Ban; Atsushi Ohno
Archive | 2014
Kazuhiro Kudou; Noriyoshi Yamamoto; Masakazu Ban; Atsushi Ohno
Archive | 2013
Noriyoshi Yamamoto; Atsushi Ohno; Kazuhiro Kudou; Masakazu Ban; Takashi Mimura; Takashi Ohtani
Archive | 2006
Masakazu Ban; Hiroshi Suhara; Masato Horiuchi; Noriyoshi Yamamoto; Hiroshi Enomoto; Hiroyuki Inoue
Archive | 2012
Kazuhiro Kudou; 一弘 工藤; Noriyoshi Yamamoto; 悟功 山本; Masakazu Ban; 正和 伴; Atsushi Ohno; 敦嗣 大野
Archive | 2006
Masakazu Ban; Hiroshi Suhara; Masato Horiuchi; Noriyoshi Yamamoto; Hiroshi Enomoto; Hiroyuki Inoue