Publication


Featured researches published by Pieter Annaert.


Drug Metabolism and Disposition | 2001

P-glycoprotein-mediated in vitro biliary excretion in sandwich-cultured rat hepatocytes

Pieter Annaert; Ryan Z. Turncliff; Catherine Booth; Dhiren R. Thakker; Kim L. R. Brouwer


Drug Metabolism and Disposition | 2004

Assessment of Drug Interactions in Hepatobiliary Transport using Rhodamine-123 in Sandwich-cultured Rat Hepatocytes

Pieter Annaert; Kim L. R. Brouwer


Archive | 2000

Modulation of p-glycoprotein (p-gp)-mediated biliary excretion in sandwich-cultured (sc) rat hepatocytes

Pieter Annaert; Edward L. LeCluyse; Kim L. R. Brouwer


Archive | 2017

Uptake, metabolism and biliary excretion of telmisartan in sandwich-cultured rat hepatocytes: comparison between freshly-isolated and cryopreserved rat hepatocytes

Neel Deferm; Janneke Keemink; Peter de Witte; Thomas Bouillon; Pieter Annaert


Archive | 2017

Modeling of telmisartan disposition in sandwich-cultured rat hepatocytes. Does cryopreservation change disposition kinetics?

Neel Deferm; Janneke Keemink; Peter de Witte; Pieter Annaert; Thomas Bouillon


Archive | 2016

Investigation of the intraluminal behavior of abiraterone acetate

Sophie Geboers; Jef Stappaerts; Raf Mols; Joachim Brouwers; Jan Tack; Jan Snoeys; Pieter Annaert; Patrick Augustijns


Archive | 2016

Pharmacokinetics, Pharmacodynamics and Drug Transport and Metabolism The Effect of Food on the Intraluminal Behavior of Abiraterone Acetate in Man

Sophie Geboers; Jef Stappaerts; Raf Mols; Jan Snoeys; Jan Tack; Pieter Annaert; Patrick Augustijns


Archive | 2016

Metabolism-based drug-drug interactions in critically ill patients: Clinical relevance & predictability of in virtro systems

Stéphane Mouly; Isabel Spriet; Joost Wauters; Pieter Annaert; Christophe Meune; Jean-François Bergmann


Archive | 2015

Transport-metabolism interplay of atazanavir in suspended rat hepatocytes

Johan Nicolaï; Tom De Bruyn; Louise Thevelin; Patrick Augustijns; Pieter Annaert


Archive | 2015

Intestinal behavior of ester prodrugs in humans: case study tenofovir DF

Sophie Geboers; Steven Haenen; Raf Mols; Joachim Brouwers; Jan Tack; Pieter Annaert; Patrick Augustijns

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