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Archive | 2017

Composés à base de 1,3-oxazin-2-amine fusionnée avec du cyclopropyle perfluoré utilisables en tant qu'inhibiteurs de la bêta-sécrétase et leurs procédés d'utilisation

Qian Wenyuan; Minatti Ana Elena; Low Jonathan D; Allen Jennifer R; Amegadzie Albert; Brown James; Frohn Michael J; Guzman-Perez Angel; Harrington Paul E; Lopez Patricia; Ma Vu Van; Nishimura Nobuko; Rumfelt Shannon; Rzasa Robert M; Sham Kelvin; Smith Adrian L; White Ryan; Xue Qiufen


Archive | 2017

PERFLUORINATED CYCLOPROPYL FUSED 1,3-OXAZIN-2-AMINE COMPOUNDS AS BETA-SECRETASE INHIBITORS AND METHODS OF USE - 13--2-

Minatti Ana Elena; Low Jonathan D; Allen Jennifer R; Amegadzie Albert; Brown James; Frohn Michael J; Guzman-Perez Angel; Harrington Paul E; Lopez Patricia; Ma Vu Van; Nishimura Nobuko; Qian Wenyuan; Rumfelt Shannon; Rzasa Robert M; Sham Kelvin; Smith Adrian L; White Ryan; Xue Qiufen


Archive | 2016

COMPUESTOS DE 1, 3-OXAZIN-2-AMINA FUSIONADOS CON CILOPROPILO PERFLUORADO COMO INHIBIDORES DE BETA-SECRETASA Y MÉTODOS DE USO

Minatti Ana Elena; Low Jonathan D; Allen Jennifer R; Amegadzie Albert; Brown James; Frohn Michael J; Guzman-Perez Angel; Harrington Paul E; Lopez Patricia; Ma Vu; Nishimura Nobuko; Qian Wenyuan; Rumfelt Shannon; Rzasa Robert M; Sham Kelvin; Smith Adrian L; White Ryan; Xue Qiufen


Archive | 2016

derivados de piridina e pirimidina como inibidores de fosfodiesterase 10

Pickrell Alex; Reichelt Andreas; Horne Daniel B; Hu Essa; Chavez Frank Junior; Demorin Frenel Fils; Yao Guomin; Monenschein Holger; Falsey James R; Allen Jennifer R; Biswas Kaustav; Sham Kelvin; Kaller Mattew R; Frohn Mike; Chen Ning; Harrington Paul; Rzasa Rob; Kunz Roxanne; Rumfelt Shannon; Nguyen Tom


Archive | 2016

ΕΝΩΣΕΙΣ ΠΥΡΑΖΙΝΗΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΦΩΣΦΟΔΙΕΣΤΕΡΑΣΗΣ 10

Allen Jennifer R; Bourbeau Matthew P; Chen Ning; Hu Essa; Kunz Roxanne; Rumfelt Shannon


Archive | 2016

composto heretocíclicos de nitrogênio úteis como inbidores pde10

Pickerell Alexander J; Harrington Essa Hu; Allen Jennifer R; Chen Jian J; Frohn Michael J; Liu Qingyian; Rzasa Robert M; Rumfelt Shannon; Zhong Wenge


Archive | 2015

Compuestos de 1,3-oxazin-2-amina fusionados con ciclopropilo perfluorado como inhibidores de beta-secretasa y métodos de uso

Minatti Ana Elena; Low Jonathan D; Allen Jennifer R; Amegadzie Albert; Brown James; Frohn Michael J; Guzman-Perez Angel; Harrington Paul E; Lopez Patricia; Ma Vu Van; Nishimura Nobuko; Qian Wenyuan; Rumfelt Shannon; Rzasa Robert M; Sham Kelvin; Smith Adrian L; White Ryan; Xue Qiufen


Archive | 2013

Compuestos heterocíclicos de nitrógeno útiles como inhibidores de pde10

Allen Jennifer R; Chen Jian J; Frohn Michael J; Harrington Essa Hu; Liu Qingyian; Pickerell Alexander J; Rumfelt Shannon; Rzasa Robert M; Zhong Wenge


Archive | 2013

Compuestos derivados de heterociclos nitrogenados insaturados o sus sales farmaceuticamente aceptables, como inhibidores de pde10; composicion farmaceutica que los comprende; y su uso para el tratamiento de enfermedades tales como psicosis, enfermedad de parkinson, depresion, trastornos del humor y demencia.

Chen Jian J; Frohn Michael J; Hu Essa; Liu Qingyian; Allen Jennifer R; Rumfelt Shannon; Rzasa Robert M; Zhong Wenge; Pickrell Alexander J


Archive | 2013

Pyrazinforbindelser som inhibitorer af Phosphodiesterase 10

Chen Ning; Hu Essa; Kunz Roxanne; Rumfelt Shannon; Allen Jennifer R; Bourbeau Matthew P

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