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Dive into the research topics where Samuel J. Gillette is active.

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Featured researches published by Samuel J. Gillette.


Archive | 2006

Pyrrolo [2, 3-b] pyridine derivatives as protein kinase inhibitors

Prabha N. Ibrahim; Dean R. Artis; Ryan Bremer; Gaston Habets; Shumeye Mamo; Marika Nespi; Chao Zhang; Jiazhong Zhang; Yong-Liang Zhu; Rebecca Zuckerman; Brian L. West; Yoshihisa Suzuki; James H. Tsai; Klaus-Peter Hirth; Gideon Bollag; Wayne Spevak; Hanna Cho; Samuel J. Gillette; Guoxian Wu; Hongyao Zhu; Shenghua Shi


Archive | 2004

Molecular scaffolds for kinase ligand development

Dean R. Artis; Ryan Bremer; Samuel J. Gillette; Clarence R. Hurt; Prabham L. Ibrahim; Rebecca Zuckerman


Archive | 2005

Bicyclic heteroaryl pde4b inhibitors

Prabham L. Ibrahim; Ryan Bremer; Samuel J. Gillette; Hanna Cho; Marika Nespi; Shumeye Mamo; Chao Zhang; Dean R. Artis; Byunghun Lee; Rebecca Zuckerman


Archive | 2010

Compounds and methods for inhibition of renin, and indications therefor

Guoxian Wu; Prabha N. Ibrahim; Yong Zhou; Shumeye Mamo; Samuel J. Gillette; Yong-Liang Zhu; Jinyu Liu; Chao Zhang; Kam Y. J. Zhang; Dean R. Artis


publisher | None

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author


Archive | 2010

Composés et procédés pour inhiber la rénine, et indications associées

Guoxian Wu; Prabha N. Ibrahim; Yong Zhou; Shumeye Mamo; Samuel J. Gillette; Yong-Liang Zhu; Jinyu Liu; Chao Zhang; Kam Y. J. Zhang; Dean R. Artis


236th National Meeting of the American-Chemical-Society | 2008

COMP 374-Potent inhibitors of mutant-B-Raf and Fms kinases designed using a scaffold-based drug discovery approach

Dean R. Artis; James H. Tsai; Ryan Bremer; Jiazhong Zhang; Hanna Cho; Shumeye Mamo; Wayne Spevak; Samuel J. Gillette; Jun Kong; Daniel Fong; Yong-Liang Zhu; Weiru Wang; Marika Nespi; Adhirai Marimuthu; Billy Lam; Shenghua Shi; Betsy Burton; Yinghui Guan; Jennifer Liu; Ivana Cheung; Julie Rice; Bernice Wong; Hoa Nguyen; Yoshihisa Suzuki; Catherine Luu; Calvin Settachatgul; Rafe Shellooe; John Cantwell; Nikolas K. Haass; Katrin Sproesser


Archive | 2006

Derives de pyrrolo [2, 3-b] pyridine utilises comme inhibiteurs de proteines kinases

Prabha N. Ibrahim; Dean R. Artis; Ryan Bremer; Gaston Habets; Shumeye Mamo; Marika Nespi; Chao Zhang; Jiazhong Zhang; Yong-Liang Zhu; Rebecca Zuckerman; Brian L. West; Yoshihisa Suzuki; James H. Tsai; Klaus-Peter Hirth; Gideon Bollag; Wayne Spevak; Hanna Cho; Samuel J. Gillette; Guoxian Wu; Hongyao Zhu; Shenghua Shi


Archive | 2006

Composes et methodes de modulation de la kinase et instructions afferentes

Prahbha N. Ibrahim; Dean R. Artis; Ryan Bremer; Shumeye Mamo; Marika Nespi; Chao Zhang; Jiazhong Zhang; Yong-Liang Zhu; James H. Tsai; Klaus-Peter Hirth; Gideon Bollag; Wayne Spevak; Hanna Cho; Samuel J. Gillette; Guoxiam Wu; Hongyao Zhu; Shenghua Shi


Archive | 2006

Pyrrolo[2,3-b]pyridin-Derivate als Proteinkinase-Hemmer

Prabha N. Ibrahim; Dean R. Artis; Ryan Bremer; Gaston Habets; Shumeye Mamo; Marika Nespi; Chao Zhang; Jiazhong Zhang; Yong-Liang Zhu; Rebecca Zuckerman; Brian L. West; Yoshihisa Suzuki; James H. Tsai; Klaus-Peter Hirth; Gideon Bollag; Wayne Spevak; Hanna Cho; Samuel J. Gillette; Guoxian Wu; Hongyao Zhu; Shenghua Shi

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