Stefano Pegoraro
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Publication
Featured researches published by Stefano Pegoraro.
Bioorganic & Medicinal Chemistry | 2009
Stefan Tasler; Oliver Müller; Tanja Wieber; Thomas Herz; Stefano Pegoraro; Wael Saeb; Martin Lang; Rolf Krauss; Frank Totzke; Ute Zirrgiebel; Jan E. Ehlert; Michael H.G. Kubbutat; Christoph Schächtele
Based on an (aminoaryl)benzothiazole quinazoline hit structure for kinase inhibition, a systematic optimization program resulted in a lead structure allowing for inhibitory activities in cellular phosphorylation assays in the low nanomolar range.
Bioorganic & Medicinal Chemistry Letters | 2009
Stefano Pegoraro; Martin Lang; Tobias Dreker; Jürgen Kraus; Svetlana Hamm; Cathal Meere; Juliane Feurle; Stefan Tasler; Sylvia Prütting; Zerrin Kuras; Violeta Visan; Stephan Grissmer
New structural classes of K(V)1.3 and IK-1 ion channel blockers have been identified based on a virtual high throughput screening approach using a homology model of KcsA. These compounds display inhibitory effects on T-cell and/or keratinocyte proliferation and immunosuppressant activity within a DTH animal model.
Archive | 2005
Johann Leban; Harald Schmitt; Kristina Wolf; Stefano Pegoraro; Andreas Wuzik
Archive | 2007
Jan Dr. Ehlert; Thomas Herz; Rolf Krauss; Michael Dr. Kubbutat; Martin Lang; Stefano Pegoraro; Christoph Schächtele; Frank Totzke; Ute Zirrgiebel
Archive | 2002
Andrea Aschenbrenner; Fuchs Katharina Aulinger; Matthias Dormeyer; Gabriel Garcia; Bernd Kramer; Juergen Kraus; Rolf Krauss; Johan Leban; Stefano Pegoraro; Wael Saeb; Kristina Wolf
Archive | 2002
Andrea Aschenbrenner; Katharina Aulinger Fuchs; Matthias Dormeyer; Gabriel Garcia; Bernd Kramer; Jürgen Kraus; Rolf Krauss; Johan Leban; Stefano Pegoraro; Wael Saeb; Kristina Wolf
Journal of Clinical Oncology | 2017
Michael Bitzer; Tom M. Ganten; Marcus A. Woerns; Jens T. Siveke; Matthias Dollinger; Max E. Scheulen; Henning Wege; Edoardo G. Giannini; Umberto Cillo; Franco Trevisani; Armando Santoro; Vincenzo Montesarchio; Anna Mais; Bernhard Hauns; Julia Asche; Thomas Herz; Stefano Pegoraro; Aldo Ammendola; Stefan W. Henning; Bernd Hentsch
Bioorganic & Medicinal Chemistry Letters | 2011
Stefano Pegoraro; Martin Lang; Tobias Dreker; Jürgen Kraus; Svetlana Hamm; Cathal Meere; Juliane Feurle; Stefan Tasler; Sylvia Prütting; Zerrin Kuras; Violeta Visan; Stephan Grissmer
Archive | 2007
Stefano Pegoraro; Martin Lang; Juliane Feurle; Juergen Krauss
Archive | 2007
Johann Leban; Harald Schmitt; Kristina Wolf; Stefano Pegoraro; Andreas Wuzik; Rolf Krauss