Takeshi Kajiwara
Takeda Pharmaceutical Company
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Publication
Featured researches published by Takeshi Kajiwara.
Catalysis Science & Technology | 2012
Takeshi Kajiwara; Takahiro Konishi; Mitsuhisa Yamano
Asymmetric catalytic hydrogenation methodology was applied to the synthesis of 2-[N-(4-difluoromethoxy)benzoylamino]cyclohexanecarboxylic acid derivatives. During the course of optimization, it was found that chiral Ru(II) dicarboxylate complexes worked efficiently with an acid additive, aqueous HBF4. Regarding chiral ligand, DTBM-BINAP showed the best result with full-conversion and the highest stereoselectivity. Practical conditions for the asymmetric hydrogenation were also established suppressing the amount of the catalyst and multi-kilogram scale synthesis was successfully achieved.
Archive | 2003
Yasushi Tanaka; Yukari Kajiwara; Makoto Noguchi; Takeshi Kajiwara; Takanori Tabuchi
Archive | 1996
Takafumi Fusaka; Osamu Ujikawa; Takeshi Kajiwara; Yasushi Tanaka
Weed Biology and Management | 2006
Yasushi Tanaka; Yukari Kajiwara; Takeshi Kajiwara; Makoto Noguchi; Naofumi Shimizu; Keizaburo Minami
Journal of Pesticide Science | 2004
Takafumi Fusaka; Seiji Yamato; Takeshi Kajiwara; Hideo Kamiyama; Shigeyuki Itoh; Yasushi Tanaka
Archive | 2003
Takanori Tabuchi; Tetsuhiro Yamamoto; Takeshi Kajiwara
Archive | 2012
Mitsuhisa Yamano; Mitsutaka Goto; Takeshi Kajiwara; Hiroyuki Maeda; Takahiro Konishi; Misayo Sera; Yuichiro Kondo; Seiji Yamasaki
Synlett | 2013
Naohiro Fukuda; Takeshi Kajiwara; Tomoaki Katou; Keisuke Majima; Tomomi Ikemoto
Archive | 2010
Takeshi Kajiwara; Satonori Tabuchi; Tetsuhiro Yamamoto; 哲寛 山本; 武志 梶原; 学典 田渕
Archive | 2005
Yasushi Tanaka; Yukari Kajiwara; Makoto Noguchi; Takeshi Kajiwara; Tabuchi Takanori