Yasunori Tsuzaki
Ube Industries
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Publication
Featured researches published by Yasunori Tsuzaki.
Bioorganic & Medicinal Chemistry Letters | 2002
Toshinori Ohmine; Tetsushi Katsube; Yasunori Tsuzaki; Miho Kazui; Nobuhiro Kobayashi; Tomoaki Komai; Masahiko Hagihara; Takashi Nishigaki; Aikichi Iwamoto; Tomio Kimura; Hiroto Kashiwase; Makoto Yamashita
Anti-HIV-1 activities and pharmacokinetics of a series of novel arylpiperazinyl fluoroquinolones are reported. Modification at the C-8 position with a trifluoromethyl group was superior to that with a difluoromethoxy group to achieve higher anti-HIV-1 activity. Two compounds studied exhibited quite high anti-HIV-1 activities (IC(50)<50 nM) in vitro and high bioavailabilities (BA>90%) in monkeys.
Archive | 1992
Hiroyuki Koike; Fumitoshi Asai; Atsuhiro Sugidachi; Tomio Kimura; Teruhiko Inoue; Shigeyoshi Nishino; Yasunori Tsuzaki
Archive | 1993
Hiroyuki Koike; Fumitoshi Asai; Atsuhiro Sugidachi; Tomio Kimura; Teruhiko Inoue; Shigeyoshi Nishino; Yasunori Tsuzaki
Archive | 2004
Masahiko Hagihara; Naoyuki Izumi; Yasunori Tsuzaki; Takeshi Matsugi; Tadashi Nakajima; Masakazu Hatano; Hideaki Hara
Archive | 2014
Kaori Taniko; Toshiyuki Miyazawa; Tatsuroh Kaneko; Daisuke Kurumazuka; Satoko Harada; Toru Izuchi; Morio Okabe; Ryo Iwamura; Yasunori Tsuzaki; Hiroyuki Setoguchi; Yuuki Imura; Hiroto Akaza; Motohisa Shimizu; Tomio Kimura
Archive | 2011
Masahiko Hagihara; Ken-Ichi Komori; Hidetoshi Sunamoto; Hiroshi Nishida; Yasunori Tsuzaki; Akira Takama; Kazutaka Kido; Tomokazu Fujimoto; Takeshi Matsugi
Archive | 1992
Hiroyuki Koike; Fumitoshi Asai; Atsuhiro Sugidachi; Tomio Kimura; Teruhiko Inoue; Shigeyoshi Nishino; Yasunori Tsuzaki
Archive | 2013
Masahiko Hagihara; Ken Komori; Hidetoshi Sunamoto; Hiroshi Nishida; Yasunori Tsuzaki; Akira Takama; Kazutaka Kido; Tomokazu Fujimoto; Takeshi Matsugi
Archive | 2011
Masahiko Hagihara; 萩原 昌彦; Ken-Ichi Komori; 健一 小森; Hidetoshi Sunamoto; 秀利 砂本; Hiroshi Nishida; 西田 洋; Yasunori Tsuzaki; 康則 津▲崎▼; Akira Takama; 昭 高間; Kazutaka Kido; 一貴 木戸; Tomokazu Fujimoto; 智和 藤本; Takeshi Matsugi; 松木 雄
Archive | 2011
Koji Ohashi; 康司 大橋; Shinichiro Hirai; 平井 慎一郎; Kazutaka Kido; 一貴 木戸; Tomokazu Fujimoto; 智和 藤本; Takeshi Matsugi; 松木 雄; Masahiko Hagihara; 萩原 昌彦; Ken-Ichi Komori; 健一 小森; Hiroshi Nishida; 西田 洋; Yasunori Tsuzaki; 康則 津▲崎▼; Akira Takama; 昭 高間