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Dive into the research topics where Hiroshi Sakashita is active.

Publication


Featured researches published by Hiroshi Sakashita.


Archive | 2001

Proline derivatives and use thereof as drugs

Hiroshi Kitajima; Hiroshi Sakashita; Fumihiko Akahoshi; Yoshiharu Hayashi


Bioorganic & Medicinal Chemistry | 2006

[(S)-γ-(Arylamino)prolyl]thiazolidine compounds as a novel series of potent and stable DPP-IV inhibitors

Hiroshi Sakashita; Fumihiko Akahoshi; Hiroshi Kitajima; Reiko Tsutsumiuchi; Yoshiharu Hayashi


Archive | 2000

Attitude determination system for artificial satellite

Shoji Yoshikawa; Katsuhiko Yamada; Hiroshi Sakashita; Hiroo Yonechi


Bioorganic & Medicinal Chemistry Letters | 2005

1-((S)-γ-Substituted prolyl)-(S)-2-cyanopyrrolidine as a novel series of highly potent DPP-IV inhibitors

Hiroshi Sakashita; Hiroshi Kitajima; Mitsuharu Nakamura; Fumihiko Akahoshi; Yoshiharu Hayashi


Bioorganic & Medicinal Chemistry | 2007

Lead optimization of [(S)-γ-(arylamino)prolyl]thiazolidine focused on γ-substituent: Indoline compounds as potent DPP-IV inhibitors

Hiroshi Sakashita; Fumihiko Akahoshi; Tomohiro Yoshida; Hiroshi Kitajima; Yoshiharu Hayashi; Shinichi Ishii; Yoko Takashina; Reiko Tsutsumiuchi; Satoshi Ono


Bioorganic & Medicinal Chemistry Letters | 2007

[(S)-γ-(4-Aryl-1-piperazinyl)-l-prolyl]thiazolidines as a novel series of highly potent and long-lasting DPP-IV inhibitors

Tomohiro Yoshida; Hiroshi Sakashita; Fumihiko Akahoshi; Yoshiharu Hayashi


Bioorganic & Medicinal Chemistry Letters | 2007

1,5-Benzodioxepin derivatives as a novel class of muscarinic M3 receptor antagonists

Shuji Sonda; Ken-ichi Katayama; Masakazu Fujio; Hiroshi Sakashita; Kenichi Inaba; Kiyoshi Asano; Toshiaki Akira


Archive | 2007

Thiazolidine derivatives and medicinal use thereof

Hiroshi Sakashita; Tomohiro Yoshida; Hiroshi Kitajima; Masahiro Takeuchi; Yoshihito Tanaka; Takuya Yoshimura; Fumihiko Akahoshi; Yoshiharu Hayashi


Archive | 1997

Lagebestimmungssystem für künstliche Satelliten

Shoji Yoshikawa; Katsuhiko Yamada; Hiroo Yonechi; Hiroshi Sakashita


Archive | 1997

Lagebestimmungssystem für künstliche Satelliten Attitude determination system for artificial satellites

Shoji Yoshikawa; Katsuhiko Yamada; Hiroo Yonechi; Hiroshi Sakashita

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