Miyasaka Tadashi
Showa University
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Publication
Featured researches published by Miyasaka Tadashi.
Biochemical Pharmacology | 1993
Baba Masanori; Yuasa Satoshi; Niwa Takuro; Yamamoto Minako; Yabuuchi Shingo; Takashima Hideaki; Ubasawa Masaru; Tanaka Hiromichi; Miyasaka Tadashi; Richard T. Walker; Jan Balzarini; Erik De Clercq; Shigeta Shiro
Several derivatives of 1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thymine (HEPT) were examined for their inhibitory effects on the replication of human immunodeficiency virus type 1 (HIV-1) in MT-4 cells in the presence of various concentrations (10-50%) of human serum (HS). Although all HEPT derivatives proved to be highly potent inhibitors of HIV-1 in the presence of 10% fetal bovine serum, some of them were less inhibitory to HIV-1 replication in the presence of HS. The HEPT derivatives were found to be highly bound to HS proteins. Both the anti-HIV-1 activity and HS protein binding of the compounds appeared to be related to their lipophilicity.
Tetrahedron | 1986
Hiromichi Tanaka; Hiroyuki Hayakawa; Kikoh Obi; Miyasaka Tadashi
Archive | 2002
Baba Masanori; Tanaka Hiromichi; Ubasawa Masaru; Walker Richard Thomas; Miyasaka Tadashi; De Clercq Erik Desire Alice; Masanori Baba
Archive | 2000
Walker Richard Thomas; Miyasaka Tadashi; Tanaka Hiromichi; De Clercq Erik Desire Alice; Baba Masanori; Ubasawa Masaru
Archive | 1999
Miyasaka Tadashi; Tanaka Hiromichi; De Clercq Erik Desire Alice; Baba Masanori; Walker Richard Thomas; Ubasawa Masaru
Archive | 1995
Miyasaka Tadashi; Tanaka Hiromichi; De Clercq Erik; Baba Masanori; Walker Richard; Ubasawa Masaru Machida Coopu
Archive | 1992
Miyasaka Tadashi; Tanaka Hiromichi; De Clerco Erik D A; Baba Masanori; Walker Richard T; Ubasawa Masaru
Archive | 1992
Miyasaka Tadashi; Tanaka Hiromichi; De Clercq Erik Desire Alice; Baba Masanori; Walker Richard Thomas; Ubasawa Masaru
Archive | 1991
Miyasaka Tadashi; Tanaka Hiromichi; De Clercq Erik Desire Alice; Baba Masanori; Walker Richard Thomas; Ubasawa Masaru
Archive | 1991
Miyasaka Tadashi; Tanaka Hiromichi; De Clercq Erik Desire Alice; Baba Masanori; Walker Richard Thomas; Ubasawa Masaru