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Dive into the research topics where Tatsuya Zenkoh is active.

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Featured researches published by Tatsuya Zenkoh.


Bioorganic & Medicinal Chemistry Letters | 2012

Discovery of novel and potent CRTH2 antagonists.

Shinji Ito; Tadashi Terasaka; Tatsuya Zenkoh; Hiroshi Matsuda; Hisashi Hayashida; Hiroshi Nagata; Yoshimasa Imamura; Miki Kobayashi; Makoto Takeuchi; Mitsuaki Ohta

High throughput screening of our chemical library for CRTH2 antagonists provided a lead compound 1a. Initial optimization of the lead led to the discovery of a novel, potent and orally bioavailable CRTH2 antagonist 17.


Archive | 1996

Benzamide derivatives and their use as vasopressin antagonists

Hiroyuki Setoi; Takehiko Ohkawa; Tatsuya Zenkoh; Hitoshi Sawada; Kentaro Sato; Hirokazu Tanaka


Archive | 1997

Benzamide derivatives having a vasopressin antagonistic activity

Hiroyuki Setoi; Takehiko Ohkawa; Tatsuya Zenkoh; Hitoshi Sawada; Yuki Sawada; Teruo Oku


Archive | 1994

Benzamide derivatives and pharmaceutical composition comprising the same

Hiroyuki Setoi; Takehiko Ohkawa; Tatsuya Zenkoh; Keiji Hemmi; Hirokazu Tanaka


Archive | 1998

QUINOLINE DERIVATIVES AS H+-ATPase INHIBITORS AND AS BONE RESORPTION INHIBITORS

Teruo Oku; Shigeki Satoh; Takayuki Inoue; Yasuharu Urano; Tatsuya Zenkoh; Noriko Yoshida


Archive | 1995

Benzamide derivatives as vasopressin antagonists

Hiroyuki Setoi; Takehiko Ohkawa; Tatsuya Zenkoh; Keiji Hemmi; Hirokazu Tanaka


Analytical Biochemistry | 2005

Selective ligand purification using high-performance affinity beads.

Yoshihiro Ohtsu; Reiko Ohba; Yoshimasa Imamura; Motoo Kobayashi; Hidetaka Hatori; Tatsuya Zenkoh; Mamoru Hatakeyama; Takashi Manabe; Motohiro Hino; Yuki Yamaguchi; Kohsuke Kataoka; Haruma Kawaguchi; Hajime Watanabe; Hiroshi Handa


Archive | 2007

Polycyclic acid compounds useful as CRTH2 antagonists and antiallergic agents

Tadashi Terasaka; Tatsuya Zenkoh; Hisashi Hayashida; Hiroshi Matsuda; Junji Sato; Yoshimasa Imamura; Hiroshi Nagata; Norio Seki; Yoshiyuki Tenda; Mamoru Tasaki; Masahiro Takeda; Seiichiro Tabuchi; Minoru Yasuda; Kazunori Tsubaki


The Journal of Antibiotics | 2003

The novel gluconeogenesis inhibitors FR225659 and FR225656 from Helicomyces sp. No. 19353. III. Structure determination.

Tatsuya Zenkoh; Yoshihiro Ohtsu; Seiji Yoshimura; Nobuharu Shigematsu; Shigehiro Takase; Motohiro Hino


Organic Letters | 2004

Design and synthesis of a solid-supported FR225659 derivative for its receptor screening

Tatsuya Zenkoh; Hidetaka Hatori; Hiroshi Tanaka; Makoto Hasegawa; Mamoru Hatakeyama; Yasuaki Kabe; Hiroyuki Setoi; Haruma Kawaguchi; Hiroshi Handa; Takashi Takahashi

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