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Dive into the research topics where Toshio Fujishita is active.

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Featured researches published by Toshio Fujishita.


Archive | 1986

Condensed imidazopyridine derivatives useful as psychotropic agents

Susumu Takada; Toshio Fujishita; Takashi Sasatani; Akira Matsushita; Masami Eigyo


Journal of Medicinal Chemistry | 1995

Novel angiotensin II receptor antagonists. Design, synthesis, and in vitro evaluation of dibenzo[a,d]cycloheptene and dibenzo[b,f]oxepin derivatives. Searching for bioisosteres of biphenylyltetrazole using a three-dimensional search technique

Ryuichi Kiyama; Tsunetoshi Honma; Kunio Hayashi; Masayoshi Ogawa; Mariko Hara; Masafumi Fujimoto; Toshio Fujishita


Journal of Medicinal Chemistry | 1980

Peptidoaminobenzophenones, a novel class of ring-opened derivatives of 1,4-benzoidazepines.

Kentaro Hirai; Teruyuki Ishiba; Hirohiko Sugimoto; Kazuyuki Sasakura; Toshio Fujishita; Tatsuro Toyoda; Yuji Tsukinoki; Hirokuni Joyama; Hisao Hatakeyama; Katsumi Hirose


Journal of Medicinal Chemistry | 1982

Amino acid amide derivatives of 2-[3-(aminomethyl)-4H-1,2,4-triazol-4-yl]benzophenones, a novel class of annelated peptidoaminobenzophenones.

Kentaro Hirai; Toshio Fujishita; Teruyuki Ishiba; Hirohiko Sugimoto; Shigeru Matsutani; Yuji Tsukinoki; Katsumi Hirose


Journal of Medicinal Chemistry | 1996

Synthesis and Structure−Activity Relationships of Fused Imidazopyridines: A New Series of Benzodiazepine Receptor Ligands

Susumu Takada; Takashi Sasatani; Nobuo Chomei; Makoto Adachi; Toshio Fujishita; Masami Eigyo; Shunji Murata; Kazuo Kawasaki; Akira Matsushita


Journal of Medicinal Chemistry | 1981

Novel peptidoaminobenzophenones, terminal N-substituted peptidoaminobenzophenones, and N-(acylglycyl)aminobenzophenones as open-ring derivatives of benzodiazepines.

Kentaro Hirai; Teruyuki Ishiba; Hirohiko Sugimoto; Toshio Fujishita; Yuji Tsukinoki; Katsumi Hirose


Chemical & Pharmaceutical Bulletin | 1995

Synthesis and Evaluation of Novel Nonpeptide Angiotensin II Receptor Antagonists : Imidazo[4, 5-c]pyridine Derivatives with an Aromatic Substituent

Ryuichi Kiyama; Masahiro Fuji; Mariko Hara; Masafumi Fujimoto; Tomoji Kawabata; Masuhisa Nakamura; Toshio Fujishita


Journal of Heterocyclic Chemistry | 1982

Synthesis and biological activity of (3,5-disubstituted-1H-1,2,4-triazol-1-yl)benzophenone derivatives †

Kentaro Hirai; Hirohiko Sugimoto; Teruyuki Ishiba; Toshio Fujishita; Yuji Tsukinoki; Katsumi Hirose


Heterocycles | 1989

Synthesis of heterocyclic compounds isosterically releated to pyrazolo[4,3-c]quinolines as benzodiazepine receptor ligands

Hirohisa Shindo; Toshio Fujishita; Takashi Sasatani; Nobuo Chomei; Susumu Takada


Chemical & Pharmaceutical Bulletin | 1978

Peptido-aminobenzophenones-Novel Open-ring Derivatives of 1,4-Benzodiazepines

Kentaro Hirai; Teruyuki Ishiba; Hirohiko Sugimoto; Kazuyuki Sasakura; Toshio Fujishita; Yuji Tsukinoki; Katsumi Hirose

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Masafumi Fujimoto

Chiba Institute of Science

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Masahiro Fuji

Kyoto Pharmaceutical University

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