Werner Zaugg
Novartis
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Publication
Featured researches published by Werner Zaugg.
Tetrahedron Letters | 2001
Olivier Lohse; Ulrich Beutler; Peter Fünfschilling; Pascal Furet; Gerhard Penn; Werner Zaugg
Abstract Benzyl and allyl protected N-o-tolyl-anthranilamides were efficiently prepared by Buchwald–Hartwig C–N cross coupling reactions, followed by protection of the amino group. Under directed remote metalation conditions, protected dibenzoazepinones were obtained in good yields. Deprotection of the amine and conversion to an urea furnished a new and efficient synthesis of the antiepileptic drug Trileptal®.
Organic Process Research & Development | 2007
Ulrich Beutler; Matthias Boehm; Peter Fuenfschilling; Thomas Heinz; Jean-Paul Mutz; Ulrich Onken; Martin Mueller; Werner Zaugg
Archive | 2003
Guang-Pei Chen; Prasad Koteswara Kapa; Eric Loeser; Ulrich Beutler; Werner Zaugg; Michael J. Girgis
Organic Process Research & Development | 2005
Peter Fuenfschilling; Werner Zaugg; Ulrich Beutler; Daniel Kaufmann; Olivier Lohse; Jean-Paul Mutz; Ulrich Onken; Jean-Louis Reber; David Shenton
Tetrahedron Letters | 2004
Peter Fünfschilling; Ulrich Beutler; Pascale Hoehn; Olivier Lohse; Werner Zaugg
Archive | 2001
Peter Fünfschilling; Daniel Kaufmann; Olivier Lohse; Ulrich Beutler; Werner Zaugg
Archive | 2001
Peter Fünfschilling; Olivier Lohse; Ulrich Beutler; Werner Zaugg
Tetrahedron Letters | 2016
Damjan Sterk; Werner Zaugg; Ulrich Beutler; Eric Loeser; Kapa Prasad; Zdenko Casar
Archive | 2009
Peter Fuenfschilling; Daniel Kaufmann; Olivier Lohse; Ulrich Beutler; Werner Zaugg
Tetrahedron Letters | 2004
Daniel Kaufmann; Peter Fünfschilling; Ulrich Beutler; Pascale Hoehn; Olivier Lohse; Werner Zaugg