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Dive into the research topics where Teresa W. Makowski is active.

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Featured researches published by Teresa W. Makowski.


Organic Process Research & Development | 2011

Use of an Iridium-Catalyzed Redox-Neutral Alcohol-Amine Coupling on Kilogram Scale for the Synthesis of a GlyT1 Inhibitor

Martin A. Berliner; Stéphane P. A. Dubant; Teresa W. Makowski; Karl Ng; Barbara J. Sitter; Carrie Wager; Yinsheng Zhang


Organic Process Research & Development | 2014

Commercial Route Research and Development for SGLT2 Inhibitor Candidate Ertugliflozin

Paul Bowles; Steven J. Brenek; Stephane Caron; Nga M. Do; Michele T. Drexler; Shengquan Duan; Pascal Dubé; Eric C. Hansen; Brian P. Jones; Kris Nicole Jones; Tomislav A. Ljubicic; Teresa W. Makowski; Jason Mustakis; Jade D. Nelson; Mark Olivier; Zhihui Peng; Hahdi H. Perfect; David William Place; John A. Ragan; John J. Salisbury; Corey L. Stanchina; Brian C. Vanderplas; Mark E. Webster; R. Matt Weekly


Journal of Organic Chemistry | 1998

SYNTHESIS OF 1,2,3,4-TETRAHYDROISOQUINOLINES CONTAINING ELECTRON-WITHDRAWING GROUPS

George J. Quallich; Teresa W. Makowski; Andrew F. Sanders; Frank J. Urban; Enrique Vazquez


Organic Process Research & Development | 2005

Investigation of Practical Routes for the Kilogram-Scale Production of cis-3-Methylamino-4-methylpiperidines

Weiling Cai; James L. Colony; Heather N. Frost; James P. Hudspeth; Peter M. Kendall; Ashwin M. Krishnan; Teresa W. Makowski; Duane J. Mazur; James Phillips; David H. Brown Ripin; Sally Gut Ruggeri; Jay F. Stearns; Timothy D. White


Organic Process Research & Development | 1998

A Practical Synthesis of Cycloheptane-1,3-dione

John A. Ragan; Teresa W. Makowski; David J. am Ende; Pamela J. Clifford; Gregory R. Young; and Alyson K. Conrad; Shane Allen Eisenbeis


Organic Letters | 2006

Enantioselective Synthesis of Nicotinic Receptor Probe 7,8-Difluoro-1,2,3,4,5,6- hexahydro-1,5-methano-3-benzazocine

Crystal G. Bashore; Michael G. Vetelino; Michael C. Wirtz; Paige R. Brooks; Heather N. Frost; Ruth E. McDermott; David C. Whritenour; John A. Ragan; Jennifer L. Rutherford; Teresa W. Makowski; and Steven J. Brenek; Jotham Wadsworth Coe


Organic Process Research & Development | 2001

Optimizing Selective Partial Hydrogenations of 4-Nitroacetophenone via Parallel Reaction Screening

Joel M. Hawkins; Teresa W. Makowski


Organic Process Research & Development | 2001

Investigation of Methods for Seven-Membered Ring Synthesis: A Practical Synthesis of 4-Oxo-5,6,7,8-tetrahydro-4H-cyclohepta[b]furan-3-carboxylic Acid

John A. Ragan; Jerry Anthony Murry; Michael J. Castaldi; Alyson Kay Conrad; Brian P. Jones; Bryan Li; Teresa W. Makowski; Ruth E. McDermott; Barb J. Sitter; and Timothy D. White; Gregory R. Young


Tetrahedron Letters | 2011

One-pot synthesis of chiral azetidines from chloroaldehyde and chiral amines

Suvi T. M. Orr; Shawn Cabral; Dilinie P. Fernando; Teresa W. Makowski


Organic Process Research & Development | 2012

Multikilogram Synthesis of a Hepatoselective Glucokinase Activator

Joshua R. Dunetz; Martin A. Berliner; Yanqiao Xiang; Timothy L. Houck; Fabrice H. Salingue; Wang Chao; Chen Yuandong; Wang Shenghua; Yun Huang; Douglas Farrand; Steven J. Boucher; David B. Damon; Teresa W. Makowski; Mark T. Barrila; Raymond Chen; Isamir Martínez

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