Zerom Tesfai
Exelixis
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Publication
Featured researches published by Zerom Tesfai.
Bioorganic & Medicinal Chemistry Letters | 2002
Adrian Folkes; S. David Brown; Lynne Canne; Jocelyn Chan; Erin Engelhardt; Sergey Epshteyn; Richard Faint; Julian Golec; Art Hanel; Patrick Kearney; James W. Leahy; Morrison B. Mac; David A. Matthews; Michael P. Prisbylla; Jason Terry Sanderson; Reyna J. Simon; Zerom Tesfai; Nigel Vicker; Shouming Wang; Robert R. Webb; Peter Charlton
We have synthesized and evaluated a series of tetramic acid-based and hydroxyquinolinone-based inhibitors of plasminogen activator inhibitor-1 (PAI-1). These studies resulted in the identification of several compounds which showed excellent potency against PAI-1. The design, synthesis and SAR of these compounds are described.
Archive | 2003
Chris A. Buhr; Tae-Gon Baik; Sunghoon Ma; Zerom Tesfai; Longcheng Wang; Erick Wang Co; Sergey Epshteyn; Abigail R. Kennedy; Baili Chen; Larisa Dubenko; Neel Kumar Anand; Tsze H. Tsang; John M. Nuss; Csaba J. Peto; Kenneth D. Rice; Mohamed Abdulkader Ibrahim; Kevin Luke Schnepp; Xian Shi; James W. Leahy; Jeff Chen; Lisa Esther Dalrymple; Thimothy Patrick Forsyth; Tai Phat Huynh; Grace Mann; Lary Wayne Mann; Craig Stacy Takeuchi
Archive | 2006
William Bajjalieh; Lynne Canne Bannen; S. David Brown; Patrick Kearney; Morrison B. Mac; Charles K. Marlowe; John M. Nuss; Zerom Tesfai; Yong Wang; Wei Xu
Archive | 2008
Suleyman Bahceci; William Bajjalieh; Jeff Chen; Sergey Epshteyn; Timothy Patrick Forsyth; Tai Phat Huynh; Byung Gyu Kim; James W. Leahy; Matthew Sangyup Lee; Gary L. Lewis; Morrison B. Mac; Grace Mann; Charles K. Marlowe; Brian Hugh Ridgway; Joan C. Sangalang; Xian Shi; Craig Stacy Takeuchi; Yong Wang; Zerom Tesfai
Archive | 2011
William Bajjalieh; Lynne Canne Bannen; S. David Brown; Patrick Kearney; Morrison B. Mac; Charles K. Marlowe; John M. Nuss; Zerom Tesfai; Yong Wang; Wei Xu
Archive | 2005
Tae-Gon Baik; Chris A. Buhr; Sunghoon Ma; John M. Nuss; Zerom Tesfai; Longcheng Wang; Bryan K. S. Yeung
Archive | 2012
Naing Aay; William Bajjalieh; Ping Huang; Lori Kabigting; Patrick Kearney; Charles K. Marlowe; Kim Moon; John M. Nuss; Arlyn Tambo-Ong; Zerom Tesfai; Amy Lew Tsuhako; Wei Xu; Christiana A. Zaharia
Archive | 2011
Neel Kumar Anand; S. David Brown; Zerom Tesfai; Cristiana A. Zaharia
Archive | 2006
William Bajjalieh; Lynne Canne Bannen; S. David Brown; Patrick Kearney; Morrison B. Mac; Charles K. Marlowe; John M. Nuss; Zerom Tesfai; Yong Wang; Wei Xu
Archive | 2006
William Bajjalieh; Bannen Lynne Canne; S. David Brown; Patrick Kearney; Morrison B. Mac; Charles K. Marlowe; John M. Nuss; Zerom Tesfai; Yong Wang; Wei Xu